EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.4.21.B25 | 0.002 |
- |
L-Arg-L-Tyr-L-Lys-L-Arg-L-Thr |
- |
707284 |
3.4.21.B25 | 0.013 |
- |
[C8]LLLLRVK-2,3-dehydroagmatine |
cell survival assay in DU145 cells, pH 7.5, 37°C |
753276 |
3.4.21.B25 | 0.015 |
- |
H2N-[C8]LLLLRVKR-NH2 |
cell survival assay in DU145 cells, pH 7.5, 37°C |
753276 |
3.4.21.B25 | 0.025 |
- |
Ac-(D)LLLLRVK-4-amidinobenzylamide |
cell survival assay in DU145 cells, pH 7.5, 37°C |
753276 |
3.4.21.B25 | 0.025 |
- |
Ac-LLLLRVK-4-amidinobenzylamide |
cell survival assay in DU145 cells, pH 7.5, 37°C |
753276 |
3.4.21.B25 | 0.03 |
- |
[C8]LLLLRVK-2,3-dehydroagmatine |
cell survival assay in LNCap cells, pH 7.5, 37°C |
753276 |
3.4.21.B25 | 0.04 |
- |
Ac-(D)LLLLRVK-2,3-dehydroagmatine |
cell survival assay in DU145 cells, pH 7.5, 37°C |
753276 |
3.4.21.B25 | 0.04 |
- |
Ac-(D)LLLLRVK-4-amidinobenzylamide |
cell survival assay in LNCap cells, pH 7.5, 37°C |
753276 |
3.4.21.B25 | 0.04 |
- |
Ac-LLLLRVK-4-amidinobenzylamide |
cell survival assay in LNCap cells, pH 7.5, 37°C |
753276 |
3.4.21.B25 | 0.04 |
- |
Ac-[C8]LLLLRVK-4-amidinobenzylamide |
cell survival assay in DU145 cells, pH 7.5, 37°C |
753276 |