EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.8.2.20 | 0.00045 |
- |
aurintricarboxylic acid |
pH 6.5, 22°C, recombinant TPST1 |
760475 |
2.8.2.20 | 0.00046 |
- |
aurintricarboxylic acid |
pH 6.5, 22°C, recombinant TPST1 |
760475 |
2.8.2.20 | 0.0005 |
- |
PSGL-1 peptide |
isoform TPST1, at pH 7.5 and 25°C |
737434 |
2.8.2.20 | 0.0007 |
- |
PSGL-1 peptide |
isoform TPST2, at pH 7.5 and 25°C |
737434 |
2.8.2.20 | 0.0014 |
- |
suramin |
pH 6.5, 22°C, recombinant TPST1 |
760475 |
2.8.2.20 | 0.0015 |
- |
adenosine 3',5'-bisphosphate |
pH 7.4, 20°C, recombinant His6-tagged enzyme |
760527 |
2.8.2.20 | 0.0016 |
- |
guanidinyl-naltrindole di-trifluoroacetate |
pH 6.5, 22°C, recombinant TPST1 |
760475 |
2.8.2.20 | 0.0024 |
- |
guanidinyl-naltrindole di-trifluoroacetate |
pH 6.5, 22°C, recombinant TPST1 |
760475 |
2.8.2.20 | 0.0065 |
- |
RAF265 |
pH 7.4, 20°C, recombinant His6-tagged enzyme |
760527 |
2.8.2.20 | 0.0099 |
- |
3'-phosphoadenosine 5'-phosphate |
isoform TPST1, at pH 7.5 and 25°C |
737434 |