EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
    2.8.2.1 | 0.00002 |
- |
2,6-Dichloro-4-nitrophenol |
isoform Sult1a1, using xanthurenic acid as substrate, in 50 mM Tris/HCl buffer, pH 7.4, 1 mM dithiothreitol, 5 mM MgCl2, and 1 mg/ml bovine serum albumin, at 37°C |
702138 |
| 2.8.2.1 | 0.00011 |
- |
meclofenamate |
pH 7.4, 37°C, versus 4-nitrophenol |
673189 |
| 2.8.2.1 | 0.00017 |
- |
2,6-Dichloro-4-nitrophenol |
isoform Sult1a1, using xanthurenic acid as substrate, in 50 mM Tris/HCl buffer, pH 7.4, 1 mM dithiothreitol, 5 mM MgCl2, and 1 mg/ml bovine serum albumin, at 37°C |
702138 |
| 2.8.2.1 | 0.00026 |
- |
4-chlorobiphenyl-3'-ol |
pH 7.0, 37°C, SULT1A1 |
673032 |
| 2.8.2.1 | 0.00039 |
- |
2,6-Dichloro-4-nitrophenol |
isoform Sult1a1, using 4-nitrophenol as substrate, in 50 mM Tris/HCl buffer, pH 7.4, 1 mM dithiothreitol, 5 mM MgCl2, and 1 mg/ml bovine serum albumin, at 37°C |
702138 |
| 2.8.2.1 | 0.0004 |
- |
2,6-Dichloro-4-nitrophenol |
isoform Sult1a1, using 4-nitrophenol as substrate, in 50 mM Tris/HCl buffer, pH 7.4, 1 mM dithiothreitol, 5 mM MgCl2, and 1 mg/ml bovine serum albumin, at 37°C |
702138 |
| 2.8.2.1 | 0.00041 |
- |
3,3',5',6-tetrachlorobiphenyl-4'-ol |
pH 7.0, 37°C, SULT1A1 |
673032 |
| 2.8.2.1 | 0.00051 |
- |
2,3,3',5,5',6-hexachlorobiphenyl-4'-ol |
pH 7.0, 37°C, SULT1A1 |
673032 |
| 2.8.2.1 | 0.00054 |
- |
2,3,3',5,6-pentachlorobiphenyl-4'-ol |
pH 7.0, 37°C, SULT1A1 |
673032 |
| 2.8.2.1 | 0.00072 |
- |
gavestinel |
isoform SULT1B1, using xanthurenic acid as substrate, in 50 mM Tris/HCl buffer, pH 7.4, 1 mM dithiothreitol, 5 mM MgCl2, and 1 mg/ml bovine serum albumin, at 37°C |
702138 |
