EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
   2.3.1.97 | -999 |
- |
more |
IC50 values of different inhibitors, overview |
720806 |
| 2.3.1.97 | 0.00000049 |
- |
(1R,3S)-N-[2-[(cyclopentylcarbonyl)amino]-1,3-benzothiazol-6-yl]-3-[(naphthalen-2-ylmethyl)amino]cyclohexanecarboxamide |
IC50: 0.00000049 mM |
672522 |
| 2.3.1.97 | 0.00000049 |
- |
(1R,3S)-N-{2-[(cyclopeanthylcarbonyl)amino]-benzothiazol-6-yl}-3-[(2-naphthylmethyl) amino] cyclohexanecarboxamide |
competitive with the substrate peptide and non-competitive with myristoyl-CoA. IC50: 0.49 nM |
672487 |
| 2.3.1.97 | 0.000001 |
- |
1-(5-[3,4-difluoro-2-[2-(1,3,5-trimethyl-1H-pyrazol-4-yl)ethoxy]phenyl]-1-methyl-1H-indazol-3-yl)-N,N-dimethylmethanamine |
IC50 value below 1 nM, pH not specified in the publication, temperature not specified in the publication |
757728 |
| 2.3.1.97 | 0.0000012 |
- |
N-[2-[(cyclopentylcarbonyl)amino]-1,3-benzothiazol-6-yl]-3-[(naphthalen-2-ylmethyl)amino]cyclohexanecarboxamide |
IC50: 0.0000012 mM |
672522 |
| 2.3.1.97 | 0.0000016 |
- |
N-[5-[(4R)-1-[(3R)-3-amino-4-(4-chlorophenyl)butanoyl]-4-(hydroxymethyl)pyrrolidin-3-yl]-2-chlorophenyl]-2-(4-fluorophenyl)acetamide |
pH not specified in the publication, temperature not specified in the publication |
736617 |
| 2.3.1.97 | 0.000002 |
- |
2,6-dichloro-4-(2-piperazin-1-ylpyridin-4-yl)-N-(1,3,5-trimethyl-1H-pyrazol-4-yl)-benzenesulfonamide |
pH 7.4, 22°C |
720195 |
| 2.3.1.97 | 0.0000023 |
- |
N-[2-[(cyclobutylcarbonyl)amino]-1,3-benzothiazol-6-yl]-3-[(naphthalen-2-ylmethyl)amino]cyclohexanecarboxamide |
IC50: 0.0000023 mM |
672522 |
| 2.3.1.97 | 0.0000024 |
- |
N-[2-[(cyclopropylcarbonyl)amino]-1,3-benzothiazol-6-yl]-3-[(naphthalen-2-ylmethyl)amino]cyclohexanecarboxamide |
IC50: 0.0000024 mM |
672522 |
| 2.3.1.97 | 0.0000033 |
- |
N-[2-[(2-methylpropanoyl)amino]-1,3-benzothiazol-6-yl]-3-[(naphthalen-2-ylmethyl)amino]cyclohexanecarboxamide |
IC50: 0.0000033 mM |
672522 |
