EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
1.2.4.1 | 0.0000026 |
- |
3-deazathiamine diphosphate |
pH 7.8, temperature not specified in the publication |
763321 |
1.2.4.1 | 0.000025 |
- |
Oxythiamine diphosphate |
pH 7.8, temperature not specified in the publication |
763321 |
1.2.4.1 | 0.0035 |
- |
N-((1-((4-amino-2-methylpyrimidin-5-yl)methyl)-5-iodo-1H-1,2,3-triazol-4-yl)methyl)-4-nitrobenzenesulfonamide |
pH 7.2, 37°C |
762797 |
1.2.4.1 | 0.0037 |
- |
N-((1-((4-amino-2-methylpyrimidin-5-yl)methyl)-5-iodo-1H-1,2,3-triazol-4-yl)methyl)-4-methoxybenzenesulfonamide |
pH 7.2, 37°C |
762797 |
1.2.4.1 | 0.0042 |
- |
5-((4-((4-bromophenoxy)methyl)-5-iodo-1H-1,2,3-triazol-1-yl)methyl)-2-methylpyrimidin-4-amine |
isolated E1 component, pH 6.5, 37°C |
758903 |
1.2.4.1 | 0.0046 |
- |
N-((1-((4-amino-2-methylpyrimidin-5-yl)methyl)-1H-1,2,3-triazol-4-yl) methyl)-2-nitrobenzenesulfonamide |
pH 7.2, 37°C |
762797 |
1.2.4.1 | 0.0051 |
- |
5-((4-((4-chloro-3-methylphenoxy)methyl)-5-iodo-1H-1,2,3-triazol-1-yl)methyl)-2-methylpyrimidin-4-amine |
isolated E1 component, pH 6.5, 37°C |
758903 |
1.2.4.1 | 0.0068 |
- |
N-((1-((4-amino-2-methylpyrimidin-5-yl)methyl)-5-iodo-1H-1,2,3-triazol-4-yl)methyl)-2,4,6-trimethylbenzenesulfonamide |
pH 7.2, 37°C |
762797 |
1.2.4.1 | 0.0071 |
- |
N-((1-((4-amino-2-methylpyrimidin-5-yl)methyl)-5-iodo-1H-1,2,3-triazol-4-yl) methyl)-4-chlorobenzenesulfonamide |
pH 7.2, 37°C |
762797 |
1.2.4.1 | 0.0078 |
- |
N-((1-((4-amino-2-methylpyrimidin-5-yl)methyl)-5-iodo-1H-1,2,3-triazol-4-yl)methyl)-4-bromobenzenesulfonamide |
pH 7.2, 37°C |
762797 |