EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
    1.14.13.9 | 0.0000003 |
- |
UPF 648 |
pH 7.4, 25°C |
725567 |
| 1.14.13.9 | 0.0000005 |
- |
6-[4-chloro-3-(cyclopropyloxy)phenyl]pyrimidine-4-carboxylic acid |
pH and temperature not specified in the publication |
764296 |
| 1.14.13.9 | 0.0000005 |
- |
6-[4-chloro-3-(cyclopropyloxy)phenyl]pyrimidine-4-carboxylic acid |
pH not specified in the publication, 37°C |
764298 |
| 1.14.13.9 | 0.0000007 |
- |
GSK366 |
pH 7.5, temperature not specified in the publication |
743342 |
| 1.14.13.9 | 0.00000071 |
- |
3-[5-(4-chloro-3-fluorophenyl)-4-methyl-1H-pyrazol-1-yl]benzoic acid |
pH 7.9, 37°C |
764520 |
| 1.14.13.9 | 0.0000013 |
- |
3-[5-chloro-2-oxo-6-[(1R)-1-(pyridazin-3-yl)ethoxy]-2,3-dihydro-1,3-benzoxazol-3-yl]propanoic acid |
pH and temperature not specified in the publication |
743067 |
| 1.14.13.9 | 0.0000014 |
- |
4-methyl-N-(6-[2-(piperidin-1-yl)phenyl]pyridazin-3-yl)benzene-1-sulfonamide |
brain enzyme, pH and temperature not specified in the publication |
764296 |
| 1.14.13.9 | 0.0000017 |
- |
4-chloro-2-([5-chloro-2-(5-methoxy-1,3-dihydro-2H-isoindol-2-yl)-1,3-thiazole-4-carbonyl](methyl)amino)-5-fluorobenzoic acid |
pH 7.9, 37°C |
764520 |
| 1.14.13.9 | 0.000002 |
- |
3-[5-chloro-2-oxo-6-[(1R)-1-(pyridin-2-yl)ethoxy]-2,3-dihydro-1,3-benzothiazol-3-yl]propanoic acid |
pH and temperature not specified in the publication |
743067 |
| 1.14.13.9 | 0.000002 |
- |
3-[5-chloro-6-[(1R)-1-(6-methylpyridazin-3-yl)ethoxy]-1,2-benzoxazol-3-yl]propanoic acid |
pH and temperature not specified in the publication |
743067 |
