EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
1.10.5.1 | 0.0000007 |
- |
S29434 |
using nicotinamide riboside and menadione as substrates, at 25°C, in 50 mM Tris-HCl, pH 8.5 |
711729 |
1.10.5.1 | 0.000005 |
- |
S29434 |
using nicotinamide riboside and coenzyme Q2 as substrates, at 25°C, in 50 mM Tris-HCl, pH 8.5 |
711729 |
1.10.5.1 | 0.000006 |
- |
5-[[4-(diethylamino)butyl]amino]-7-hydroxy-8,9-dimethoxy-6H-imidazo[4,5,1-de]acridin-6-one |
pH and temperature not specified in the publication |
711408 |
1.10.5.1 | 0.000006 |
- |
NSC660841 |
pH and temperature not specified in the publication |
711408 |
1.10.5.1 | 0.0000067 |
- |
S29434 |
using N-benzyl dihydronicotinamide and menadione as substrates, at 25°C, in 50 mM Tris-HCl, pH 8.5 |
711729 |
1.10.5.1 | 0.000009 |
- |
5-[[4-(diethylamino)butyl]amino]-8-methoxy-1-methyl-6H-imidazo[4,5,1-de]acridin-6-one |
pH and temperature not specified in the publication |
711408 |
1.10.5.1 | 0.000009 |
- |
NSC637993 |
pH and temperature not specified in the publication |
711408 |
1.10.5.1 | 0.000014 |
- |
N-[2-(2-methoxy-6H-dipyrido[2,3-a:3,2-e]pyrrolizin-11-yl)ethyl]-2-furamide |
IC50: 14 nM |
657889 |
1.10.5.1 | 0.000016 |
- |
5-[[4-(diethylamino)butyl]amino]-8-hydroxy-1-methyl-6H-imidazo[4,5,1-de]acridin-6-one |
pH and temperature not specified in the publication |
711408 |
1.10.5.1 | 0.000016 |
- |
chrysoeriol |
using nicotinamide riboside and menadione as substrates, at 25°C, in 50 mM Tris-HCl, pH 8.5 |
711729 |