EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference  |
|---|
    4.4.1.20 | 0.06 |
- |
Sulfobromophthalein |
IC50: 0.06 mM |
644509 |
| 4.4.1.20 | 0.26 |
- |
p-aminohippuric acid |
IC50: 0.26 mM |
644509 |
| 4.4.1.20 | 1.9 |
- |
estrone-3-sulfate |
IC50: 1.9 mM |
644509 |
| 4.4.1.20 | 17 |
- |
probenecid |
IC50: 17 mM |
644509 |
| 4.4.1.20 | 0.000135 |
- |
2-benzoyl-5-(5-[(4-chlorophenyl)(methyl)amino]pyridine-2-carbonyl)benzoic acid |
pH 7.8, temperature not specified in the publication, recombinant enzyme |
730788 |
| 4.4.1.20 | 0.000017 |
- |
5-[5-[(4-chlorophenyl)(methyl)amino]pyridine-2-carbonyl]-2-(4-methoxybenzoyl)benzoic acid |
cell-free assay, the substrate LTA4 is produced in situ, 37°C, pH not specified in the publication |
747181 |
| 4.4.1.20 | 0.000095 |
- |
5-[5-[(4-chlorophenyl)(cyclopropylmethyl)amino]pyridine-2-carbonyl]-2-(4-methoxybenzoyl)benzoic acid |
pH not specified in the publication, temperature not specified in the publication |
748456 |
| 4.4.1.20 | 0.000116 |
- |
2-benzoyl-5-[5-[(4-chlorophenyl)(methyl)amino]pyridine-2-carbonyl]benzoic acid |
pH not specified in the publication, temperature not specified in the publication |
748456 |
| 4.4.1.20 | 0.000124 |
- |
5-[5-[(4-chlorophenyl)(methyl)amino]pyridine-2-carbonyl]-2-(4-methoxybenzoyl)benzoic acid |
pH not specified in the publication, temperature not specified in the publication |
748456 |
