EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
   3.6.4.10 | 0.0046 |
- |
8-(2-chloro-3,4,5-trimethoxybenzyl)-2-fluoro-9-(pent-4-yn-1-yl)-9H-purin-6-amine |
pH and temperature not specified in the publication |
719075 |
| 3.6.4.10 | 0.0089 |
- |
4-[4-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-1H-pyrazol-3-yl]-6-ethylbenzene-1,3-diol |
pH and temperature not specified in the publication |
719075 |
| 3.6.4.10 | 0.0309 |
- |
17-allylamino-17-demethoxygeldanamycin |
inhibition of the ATPase activity, pH 7.4, temperature not specified in the publication |
734478 |
| 3.6.4.10 | 0.065 |
- |
5-[1-[(6-[5-[(benzyloxy)carbonyl]-4-biphenyl-4-yl-6-methyl-2-oxo-3,4-dihydropyrimidin-1(2H)-yl]hexanoyl)(hexyl)amino]-2-[(1E)-butylideneamino]-2-oxoethyl]-2-(carboxymethoxy)benzoic acid |
pH 7.4, 37°C, presence of peptide NRLLLTG |
684406 |
| 3.6.4.10 | 0.115 |
- |
17-allylamino-17-demethoxygeldanamycin |
inhibition of the ATPase activity, in presence of co-chaperone EhAha1c, pH 7.4, temperature not specified in the publication |
734478 |
| 3.6.4.10 | 0.13 |
- |
5-[1-[(6-[5-[(benzyloxy)carbonyl]-4-biphenyl-4-yl-6-methyl-2-oxo-3,4-dihydropyrimidin-1(2H)-yl]hexanoyl)(hexyl)amino]-2-[(1E)-butylideneamino]-2-oxoethyl]-2-(carboxymethoxy)benzoic acid |
pH 7.4, 37°C |
684406 |
