EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
3.5.1.60 | 0.1 |
- |
methyl 3-[7-oxo-7-(pyrrolidin-1-yl)heptyl]benzoate |
above, pH 4.5, 37°C |
754610 |
3.5.1.60 | 0.1 |
- |
methyl 4-[7-oxo-7-(pyrrolidin-1-yl)heptyl]benzoate |
above, pH 4.5, 37°C |
754610 |
3.5.1.60 | 0.1 |
- |
N-pentadecylnaphthalene-2-carboxamide |
above, pH and temperature not specified in the publication |
752960 |
3.5.1.60 | 0.1 |
- |
N-[(2R,3S)-2-methyl-4-oxooxetan-3-yl]-3-phenylpropanamide |
above, pH and temperature not specified in the publication |
734845 |
3.5.1.60 | 0.44 |
- |
3-[6-(4-methylphenyl)hexanoyl]-1,3-oxazolidin-2-one |
above, pH and temperature not specified in the publication |
753491 |
3.5.1.60 | 0.48 |
- |
3-(4-phenylcyclohexyl)-1-(pyrrolidin-1-yl)propan-1-one |
pH 4.5, 37°C |
754610 |
3.5.1.60 | 1.5 |
- |
(2E)-3-([1,1'-biphenyl]-4-yl)-1-(pyrrolidin-1-yl)prop-2-en-1-one |
pH 4.5, 37°C |
754610 |
3.5.1.60 | 2.8 |
- |
3-(4-phenoxycyclohexyl)-1-(pyrrolidin-1-yl)propan-1-one |
pH 4.5, 37°C |
754610 |
3.5.1.60 | 4.1 |
- |
(2E,4E)-5-(2H-1,3-benzodioxol-5-yl)-1-(pyrrolidin-1-yl)penta-2,4-dien-1-one |
pH 4.5, 37°C |
754610 |
3.5.1.60 | 5.5 |
- |
5-(2H-1,3-benzodioxol-5-yl)-1-(pyrrolidin-1-yl)pentan-1-one |
pH 4.5, 37°C |
754610 |