EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
   3.4.22.69 | 0.03857 |
- |
N-[(1Z)-3-[[3-(dimethylamino)propyl]amino]-1-[5-(3-nitrophenyl)furan-2-yl]-3-oxoprop-1-en-2-yl]-4-methylbenzamide |
pH and temperature not specified in the publication |
717343 |
| 3.4.22.69 | 0.04 |
- |
2-(4,5-dihydro-1,3-thiazol-2-yl)-1-(1,3-thiazol-2-yl)ethanone |
- |
681289 |
| 3.4.22.69 | 0.04 |
- |
3-[N-(N-tert-butoxycarbonyl)-L-Leu]-1,1,1-trifluorobutan-2-one |
- |
691222 |
| 3.4.22.69 | 0.04 |
- |
3-[N-[N-tert-butoxycarbonyl-L-gamma-Glu(OtBu)-L-Ala]]-1,1,1-trifluoropropan-2-one |
- |
691222 |
| 3.4.22.69 | 0.04 |
- |
curcumin |
- |
681313 |
| 3.4.22.69 | 0.04 |
- |
niclosamide |
- |
681313 |
| 3.4.22.69 | 0.041 |
- |
(2S)-2-([[(3S,4aR,8aS)-2-(4-bromobenzoyl)decahydroisoquinolin-3-yl]methyl]amino)-3-(1H-imidazol-4-yl)propanal |
pH 7.5, 37°C |
752951 |
| 3.4.22.69 | 0.04139 |
- |
N-[(1Z)-3-[[3-(dimethylamino)propyl]amino]-1-[5-(2-nitrophenyl)furan-2-yl]-3-oxoprop-1-en-2-yl]-4-methylbenzamide |
pH and temperature not specified in the publication |
717343 |
| 3.4.22.69 | 0.043 |
- |
(S)-N-((S)-1-(benzo[d]thiazol-2-yl)-1-oxo-3-((S)-2-oxopyrrolidin-3-yl)propan-2-yl)-2-(2-(4-methoxyphenyl)acetamido)-4-methylpentanamide |
enzyme mutant R188I, pH and temperature not specified in the publication |
731748 |
| 3.4.22.69 | 0.043 |
- |
1,6-di(propan-2-yl)-N-(4-[[4-(prop-2-en-1-yl)-5-sulfanylidene-4,5-dihydro-1H-1,2,4-triazol-3-yl]methyl]-1,3-thiazol-2-yl)-1H-pyrazolo[3,4-b]pyridine-4-carboxamide |
mutant R188I, pH not specified in the publication, temperature not specified in the publication |
752992 |
