EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
   3.4.22.69 | 0.025 |
- |
1,1'-sulfonylbis(4-nitrobenzene) |
- |
681289 |
| 3.4.22.69 | 0.025 |
- |
savinin |
- |
681313 |
| 3.4.22.69 | 0.0253 |
- |
2-(1H-benzotriazol-1-yl)-N-[2-(tert-butylamino)-2-oxo-1-(thiophen-3-yl)ethyl]-N-[4-[(methylsulfonyl)amino]phenyl]acetamide |
pH and temperature not specified in the publication |
731443 |
| 3.4.22.69 | 0.026 |
- |
acetyl-Thr-Ser-Ala-Val-Leu-NHCH(CH2CH2CON(CH3)2)-CHO |
- |
691242 |
| 3.4.22.69 | 0.026 |
- |
N-(4-[(1H-benzotriazol-1-ylacetyl)[2-(tert-butylamino)-2-oxo-1-(thiophen-3-yl)ethyl]amino]phenyl)-1,2-oxazole-5-carboxamide |
pH and temperature not specified in the publication |
731443 |
| 3.4.22.69 | 0.026 |
- |
N-acetyl-L-threonyl-N-[(3R,4S,4aR,8aS)-2-(4-bromobenzoyl)-3-([[(2S)-1-(1H-imidazol-4-yl)-3-oxopropan-2-yl]amino]methyl)decahydroisoquinolin-4-yl]glycinamide |
pH 7.5, 37°C |
752974 |
| 3.4.22.69 | 0.0263 |
- |
4-(4-methoxyphenyl)-2-[(4-nitrobenzyl)sulfanyl]-6-oxo-1,6-dihydropyrimidine-5-carbonitrile |
- |
707708 |
| 3.4.22.69 | 0.028 |
- |
2-(5-bromopyridin-3-yl)-1-(5-(4-chlorophenyl)furan-2-yl)-2-fluoroethanone |
- |
691200 |
| 3.4.22.69 | 0.03 |
- |
(R)-N-cinnamoyl serine(benzoyl)cyclohexylamide |
pH 4.0, temperature not specified in the publication |
752992 |
| 3.4.22.69 | 0.0318 |
- |
tafenoquine |
pH 7.8, 25°C |
765085 |
