EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.7.11.10 | 0.0083 |
- |
N-(6-chloro-9H-beta-carbolin-8-yl)methanesulfonamide |
inhibits IKK with IC50 of 0.0083 mM |
661333 |
2.7.11.10 | 0.0085 |
- |
3-amino-6-methyl-4-(4-methylphenyl)thieno[2,3-b]pyridine-2-carboxamide |
IKKbeta |
702590 |
2.7.11.10 | 0.0085 |
- |
4-(1-benzothiophen-2-yl)-N-[4-(pyrrolidin-1-ylcarbonyl)phenyl]pyrimidin-2-amine |
IC50 for the IKK complex is 0.0085 mM, cellular profile |
661346 |
2.7.11.10 | 0.0086 |
- |
ethanol,N-[2-[[2-(4-fluorophenyl)-8-methyl-8H-imidazo[4,5-d]thiazolo[5,4-b]pyridine-5-yl]amino]ethyl] |
IKK-1 |
705026 |
2.7.11.10 | 0.0097 |
- |
N-[5-[4-(cyclopropylamino)-1-methyl-1H-pyrazolo[5,1-b]purin-7-yl]-2-fluorobenzyl]acetamide |
IKK-1 |
705026 |
2.7.11.10 | 0.0098 |
- |
2-amino-4-(3-(hydroxymethyl)phenyl)-7H-pyrrolo[2,3-d]-pyrimidine-5-carbonitrile |
at pH 7.5 and 30°C |
761671 |
2.7.11.10 | 0.0098 |
- |
3-amino-6-(4-hydroxypiperidin-1-yl)-4-propylthieno[2,3-b]pyridine-2-carboxamide |
whole blood assay |
702590 |
2.7.11.10 | 0.01 |
- |
2-amino-4-(4-fluorophenyl)-7H-pyrrolo[2,3-d]pyrimidine-5-carbonitrile |
at pH 7.5 and 30°C |
761671 |
2.7.11.10 | 0.01 |
- |
4-((2-amino-5-cyano-7H-pyrrolo[2,3-d]pyrimidin-4-yl)amino)-benzenesulfonamide |
at pH 7.5 and 30°C |
761671 |
2.7.11.10 | 0.01 |
- |
6-bromo-7-(piperidin-4-yloxy)isoquinoline |
IKK-alpha |
705033 |