EC Number   |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
|---|
    2.4.2.30 | 0.294 |
- |
3-(4-methoxy-6,7-dihydro-5H-cyclopenta[4,5]thieno[2,3-d]pyrimidin-2-yl)propanoic acid |
at pH 7.5 and 22°C |
736518 |
| 2.4.2.30 | 0.003 |
- |
4-nitro-7-[(1-oxo-1lambda(5)-pyridin-2-yl)sulfanyl]-2,1,3-benzoxadiazole |
at pH 7.5 and 25°C |
758573 |
| 2.4.2.30 | 0.0068 |
- |
4,5,7,9-tetrahydro-2H-purine-2,8(3H)-dithione |
at pH 7.5 and 25°C |
758573 |
| 2.4.2.30 | 0.02 |
- |
(1E,4E)-1,5-di(pyridin-3-yl)penta-1,4-dien-3-one |
at pH 7.5 and 25°C |
758573 |
| 2.4.2.30 | 0.22 |
- |
3-amino-1,4-dimethyl-5H-pyrido[4,3-b]indole |
i.e. Trp-P-1, 94% inhibition at 5 mM, IC50: 0.22 mM |
675627 |
| 2.4.2.30 | 2.2 |
- |
3-amino-1-methyl-5H-pyrido[4,3-b]indole |
i.e. Trp-P-2, 34% activation at 1 mM, 7% inhibition at 5 mM, IC50: 2.2 mM |
675627 |
| 2.4.2.30 | 0.1 |
- |
3-(4-oxo-3,4-dihydroquinazolin-2-yl)-N-[(1R)-1-(pyridin-2-yl)ethyl]propanamide |
IC50 above 0.1 mM, pH and temperature not specified in the publication |
736615 |
| 2.4.2.30 | 0.1 |
- |
N-[(1R)-2,3-dihydro-1H-inden-1-yl]-3-(4-oxo-3,4-dihydroquinazolin-2-yl)propanamide |
IC50 above 0.1 mM, pH and temperature not specified in the publication |
736615 |
| 2.4.2.30 | 0.1 |
- |
N-[(1S)-2,3-dihydro-1H-inden-1-yl]-3-(4-oxo-3,4-dihydroquinazolin-2-yl)propanamide |
IC50 above 0.1 mM, pH and temperature not specified in the publication |
736615 |
| 2.4.2.30 | 0.00018 |
- |
4-amino-1,8-naphthalimide |
IC50: 0.00018 mM |
637997 |
