EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
6.1.1.18 | 0.06 |
- |
I- |
- |
114 |
6.1.1.18 | 0.1 |
- |
Br- |
- |
114 |
6.1.1.18 | 0.2 |
- |
Cl- |
- |
114 |
6.1.1.18 | -999 |
- |
more |
inhibition kinetics |
672564 |
6.1.1.18 | 29 |
- |
L-Glutamic acid |
mutant F90L, pH 7.2, 37°C |
651246 |
6.1.1.18 | 21 |
- |
L-Glutamic acid |
mutant Y240E, pH 7.2, 37°C |
651246 |
6.1.1.18 | 47 |
- |
L-Glutamic acid |
mutant Y240G, pH 7.2, 37°C |
651246 |
6.1.1.18 | 0.0013 |
- |
5'-O-[N-(L-glutaminyl)sulfamoyl] adenosine |
pH 7.0, 37°C |
653922 |
6.1.1.18 | 0.65 |
- |
glutaminyl-beta-ketophosphonate-adenosine |
pH 7.2, 37°C, versus L-glutamine |
672564 |
6.1.1.18 | 2.8 |
- |
glutamyl-beta-ketophosphonate-adenosine |
pH 7.2, 37°C, versus L-glutamine |
672564 |