EC Number   |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
|---|
   5.2.1.8 | 0.000001 |
- |
(3S,26aR)-19,19-dimethyl-3-(2-phenylethyl)-12,13,14,15,18,19,24,25,26,26a-decahydro-3H,10H-4,8-(metheno)pyrido[2,1-c][1,9,17,4]trioxazacyclotricosine-1,16,20,21(11H,23H)-tetrone |
- |
680340 |
| 5.2.1.8 | 0.0000028 |
- |
benzyl (2S)-1-[[(1S,2R,5R)-1-hydroxy-5-[(1S)-1-methoxy-3-methylbutyl]-2-methylcyclohexyl](oxo)acetyl]piperidine-2-carboxylate |
- |
678717 |
| 5.2.1.8 | 0.0000039 |
- |
cyclosporin A |
- |
653459 |
| 5.2.1.8 | 0.000005 |
- |
(1R)-1-[3-(diethenylcarbamoyl)phenyl]-3-phenylpropyl 1-(3,3-dimethyl-2-oxopentanoyl)piperidine-2-carboxylate |
- |
678715 |
| 5.2.1.8 | 0.000005 |
- |
(1R)-3-phenyl-1-[3-(phenylcarbonyl)phenyl]propyl 1-(3,3-dimethyl-2-oxopentanoyl)piperidine-2-carboxylate |
- |
678715 |
| 5.2.1.8 | 0.000007 |
- |
(1S)-1-cyclohexyl-3-phenylpropyl (2R)-1-(3,3-dimethyl-2-oxopentanoyl)piperidine-2-carboxylate |
- |
680340 |
| 5.2.1.8 | 0.00001 |
- |
(1R)-1,3-diphenyl-1-propyl (2S)-1-(3,3-dimethyl-1,2-dioxopentyl)-2-piperidinecarboxylate |
- |
680340 |
| 5.2.1.8 | 0.000012 |
- |
3-(3,4,5-trimethoxyphenyl)propyl (2R)-1-(3,3-dimethyl-2-oxopentanoyl)piperidine-2-carboxylate |
- |
680340 |
| 5.2.1.8 | 0.0000188 |
- |
cyclosporin A |
pH 8.0, 15°C |
749062 |
| 5.2.1.8 | 0.000019 |
- |
4-phenyl-1-(3-pyridin-3-ylpropyl)butyl (2R)-1-[difluoro(3,4,5-trimethoxyphenyl)acetyl]piperidine-2-carboxylate |
- |
682235 |
