EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.5.1.98 | 0.0007 |
- |
7-mercapto-N-phenylheptanamide |
- |
681276 |
3.5.1.98 | 0.046 |
- |
Butyrate |
- |
697650 |
3.5.1.98 | 0.0085 |
- |
N-hydroxy-1-methyl-indole-6-carboxamide |
HDAC1 inhibition |
697087 |
3.5.1.98 | 0.000015 |
- |
PCI-34051 |
HDAC8 inhibition |
697087 |
3.5.1.98 | 0.0007 |
- |
(2E)-N-hydroxy-3-naphthalen-1-ylprop-2-enamide |
HDAC8 inhibition |
697087 |
3.5.1.98 | 0.0013 |
- |
N-hydroxy-1-methyl-indole-6-carboxamide |
HDAC8 inhibition |
697087 |
3.5.1.98 | 0.014 |
- |
N-hydroxynaphthalene-1-carboxamide |
HDAC8 inhibition |
697087 |
3.5.1.98 | 0.0000137 |
- |
methyl (3R,6R,9R)-9-(acetylamino)-6-[6-(hydroxyamino)-6-oxohexyl]-5,8-dioxo-4,7-diazabicyclo[9.3.1]pentadeca-1(15),11,13-triene-3-carboxylate |
HeLa cell nuclear extract |
681304 |
3.5.1.98 | 0.024 |
- |
allyl mercaptan |
human HDAC8 |
697650 |
3.5.1.98 | -999 |
- |
more |
inhibition kinetic calculations, Kd values, detailed overview |
733081 |