EC Number   |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
|---|
   3.4.23.5 | 0.0000005 |
- |
pepstatin A |
pH 2.2, 30°C |
650901 |
| 3.4.23.5 | 0.0000007 |
- |
pyridine-2-carboxylic acid ((S)-1-((1S,2S)-1-(4-benzo-[1,3]dioxol-5-yl-benzyloxymethyl)-3-[(S)-1-((S)-1-carbamoyl-3-methyl-butylcarbamoyl)-ethylcarbamoyl]-2-hydroxypropylcarbamoyl)-2-methylpropyl)-amide |
- |
669779 |
| 3.4.23.5 | 0.0000016 |
- |
pyridine-2-carboxylic acid ((S)-1-[(1S,2S)-3-[(S)-1-((S)-1-carbamoyl-3-methylbutylcarbamoyl)-ethylcarbamoyl]-2-hydroxy-1-(3-thiophen-3-yl-benzyloxymethyl)-propylcarbamoyl]-2-methyl-propyl)-amide |
- |
669779 |
| 3.4.23.5 | 0.0000025 |
- |
pyridine-2-carboxylic acid ((S)-1-((1S,2S)-1-(biphenyl-4-ylmethoxymethyl)-3-[(S)-1-((S)-1-carbamoyl-3-methyl-butylcarbamoyl)-ethylcarbamoyl]-2-hydroxy-propylcarbamoyl)-2-methyl-propyl)-amide |
- |
669779 |
| 3.4.23.5 | 0.0000027 |
- |
pepstatin A |
40°C, pH 4.0, gastric cathepsin D, hydrolysis of (7-methoxycoumarin-4-yl)acetyl-Gly-Ser-Pro-Ala-Phe-Leu-Ala-Lys(Dnp)-D-Arg-NH2 |
667861 |
| 3.4.23.5 | 0.00000307 |
- |
pepstatin A |
in 0.05 M sodium acetate buffer, pH 3.5, at 45°C |
718074 |
| 3.4.23.5 | 0.0000031 |
- |
pepstatin A |
40°C, pH 4.0, spleen cathepsin D, hydrolysis of (7-methoxycoumarin-4-yl)acetyl-Gly-Ser-Pro-Ala-Phe-Leu-Ala-Lys(Dnp)-D-Arg-NH2 |
667861 |
| 3.4.23.5 | 0.0000032 |
- |
cathepsin D inhibitor from Streptomyces sp.MBR04 |
in 0.02M sodium citrate, pH 3.0, at 37°C |
731168 |
| 3.4.23.5 | 0.0000032 |
- |
pyridine-2-carboxylic acid ((S)-1-[(1S,2S)-3-[(S)-1-((S)-1-carbamoyl-3-methyl-butylcarbamoyl)-ethylcarbamoyl]-2-hydroxy-1-(4-thiophen-3-yl-benzyloxymethyl)-propyl-carbamoyl]-2-methyl-propyl)-amide |
- |
669779 |
| 3.4.23.5 | 0.0000039 |
- |
pyridine-2-carboxylic acid ((S)-1-((1S,2S)-1-(biphenyl-3-ylmethoxymethyl)-3-[(S)-1-((S)-1-carbamoyl-3-methyl-butylcarbamoyl)-ethylcarbamoyl]-2-hydroxy-propylcar-bamoyl)-2-methyl-propyl)-amide |
- |
669779 |
