EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.4.23.24 | -999 |
- |
more |
second order inhibition rate constants between 56.000 and 121.000M(-1)min(-1) for cis-configured epoxides and aziridines |
679234 |
3.4.23.24 | 0.00000003 |
- |
benzyloxycarbonyl-L-Val-L-Val-statine-L-Ala-statine-OH |
isoform Sapp2p, in 150 mM sodium citrate buffer, pH 3.75, at 37°C |
707611 |
3.4.23.24 | 0.0000001 |
- |
benzyloxycarbonyl-L-Val-L-Val-((3S,4S)-4-amino-3-hydroxy-5-phenylpentanoic acid)-L-Ala-((3R,4R)-4-amino-3-hydroxy-5-phenylpentanoic acid)-OMe |
isoform Sapp2p, in 150 mM sodium citrate buffer, pH 3.75, at 37°C |
707611 |
3.4.23.24 | 0.0000001 |
- |
benzyloxycarbonyl-L-Val-L-Val-((3S,4S)-4-amino-3-hydroxy-5-phenylpentanoic acid)-L-Ala-((3S,4S)-4-amino-3-hydroxy-5-phenylpentanoic acid)-NH2 |
isoform Sapp1p, in 150 mM sodium citrate buffer, pH 3.75, at 37°C |
707611 |
3.4.23.24 | 0.0000001 |
- |
benzyloxycarbonyl-L-Val-L-Val-((3S,4S)-4-amino-3-hydroxy-5-phenylpentanoic acid)-L-Ala-((3S,4S)-4-amino-3-hydroxy-5-phenylpentanoic acid)-NH2 |
isoform Sapp2p, in 150 mM sodium citrate buffer, pH 3.75, at 37°C |
707611 |
3.4.23.24 | 0.0000002 |
- |
benzyloxycarbonyl-L-Val-L-Val-((3S,4S)-4-amino-3-hydroxy-5-phenylpentanoic acid)-L-Ala-( (3S,4S)-4-amino-3-hydroxy-5-phenylpentanoic acid)-OMe |
isoform Sapp2p, in 150 mM sodium citrate buffer, pH 3.75, at 37°C |
707611 |
3.4.23.24 | 0.0000003 |
- |
benzyloxycarbonyl-L-Val-L-Val-((3S,4S)-4-amino-3-hydroxy-5-phenylpentanoic acid)-L-Ala-( (3S,4S)-4-amino-3-hydroxy-5-phenylpentanoic acid)-OMe |
isoform Sapp1p, in 150 mM sodium citrate buffer, pH 3.75, at 37°C |
707611 |
3.4.23.24 | 0.0000003 |
- |
benzyloxycarbonyl-L-Val-L-Val-statine-L-Ala-statine-OH |
isoform Sapp1p, in 150 mM sodium citrate buffer, pH 3.75, at 37°C |
707611 |
3.4.23.24 | 0.0000003 |
- |
isovaleryl-Val-Val-statyl-Ala-statyl-OH |
- |
667864 |
3.4.23.24 | 0.0000003 |
- |
pepstatin A |
isoform Sapp1p, in 150 mM sodium citrate buffer, pH 3.75, at 37°C |
707611 |