EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.4.22.62 | 0.0142 |
- |
benzyloxycarbonyl-VAE-fluoromethylketone |
- |
666835 |
3.4.22.62 | 0.0171 |
- |
benzyloxycarbonyl-VAD-fluoromethylketone |
- |
666835 |
3.4.22.62 | 0.0015 |
- |
Zn2+ |
mutant C172A, pH 6.5, 37°C |
732880 |
3.4.22.62 | 0.0012 |
- |
Zn2+ |
mutant C239S, pH 6.5, 37°C |
732880 |
3.4.22.62 | 0.0007 |
- |
Zn2+ |
mutant C272A, pH 6.5, 37°C |
732880 |
3.4.22.62 | 0.0002 |
- |
Zn2+ |
mutant C272A/C287A, pH 6.5, 37°C |
732880 |
3.4.22.62 | 0.0008 |
- |
Zn2+ |
mutant C287A, pH 6.5, 37°C |
732880 |
3.4.22.62 | 0.0007 |
- |
Zn2+ |
mutant C287A/C239S, pH 6.5, 37°C |
732880 |
3.4.22.62 | 0.0008 |
- |
Zn2+ |
mutant H237A, pH 6.5, 37°C |
732880 |
3.4.22.62 | 0.000048 |
- |
acetyl-AEVD-CHO |
pH 7.5, 25°C |
647423 |