EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.4.21.B25 | 0.0000007 |
- |
Ac-[PEG8]LLLLRVK-4-amidinobenzylamide |
pH 7.5, 37°C |
753276 |
3.4.21.B25 | 0.000001 |
- |
H2N-[C8]LLLLRVK-4-amidinobenzylamide |
pH 7.5, 37°C |
753276 |
3.4.21.B25 | 0.0000027 |
- |
Ac-[PEG2](D)LLLLRVK-4-amidinobenzylamide |
pH 7.5, 37°C |
753276 |
3.4.21.B25 | 0.0000028 |
- |
Ac-[PEG8]LLLLRVK-2,3-dehydroagmatine |
pH 7.5, 37°C |
753276 |
3.4.21.B25 | 0.0000029 |
- |
Ac-[PEG8](D)LLLLRVK-4-amidinobenzylamide |
pH 7.5, 37°C |
753276 |
3.4.21.B25 | 0.000003 |
- |
Ac-[C8]LLLLRVK-4-amidinobenzylamide |
pH 7.5, 37°C |
753276 |
3.4.21.B25 | 0.0000031 |
- |
Ac-LLLLRVK-4-amidinobenzylamide |
pH 7.5, 37°C |
753276 |
3.4.21.B25 | 0.0000034 |
- |
H2N-[C8]LLLLRVK-2,3-dehydroagmatine |
pH 7.5, 37°C |
753276 |
3.4.21.B25 | 0.0000045 |
- |
H2N-[C8](D)LLLLRVK-2,3-dehydroagmatine |
pH 7.5, 37°C |
753276 |
3.4.21.B25 | 0.0000049 |
- |
Ac-(D)LLLLRVK-4-amidinobenzylamide |
pH 7.5, 37°C |
753276 |