EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.4.15.1 | 100 |
- |
PO43- |
- |
81286 |
3.4.15.1 | 500 |
- |
NaCl |
- |
81286 |
3.4.15.1 | 0.000009 |
- |
captopril |
pH 8.0, 37°C, N-domain, hydrolysis of o-aminobenzoyl-SDK-(dinitrophenyl)-P-OH |
650001 |
3.4.15.1 | 0.00001 |
- |
captopril |
pH 8.0, 37°C, wild-type enzyme, hydrolysis of o-aminobenzoyl-SDK-(dinitrophenyl)-P-OH |
650001 |
3.4.15.1 | 0.000016 |
- |
captopril |
pH 8.0, 37°C, C-domain, hydrolysis of o-aminobenzoyl-FRK-(dinitrophenyl)-P-OH |
650001 |
3.4.15.1 | 0.000025 |
- |
captopril |
pH 8.0, 37°C, N-domain, hydrolysis of o-aminobenzoyl-FRK-(dinitrophenyl)-P-OH |
650001 |
3.4.15.1 | 0.000046 |
- |
captopril |
pH 8.0, 37°C, wild-type enzyme, hydrolysis of o-aminobenzoyl-FRK-(dinitrophenyl)-P-OH |
650001 |
3.4.15.1 | 0.000191 |
- |
captopril |
pH 8.0, 37°C, C-domain, hydrolysis of o-aminobenzoyl-SDK-(dinitrophenyl)-P-OH |
650001 |
3.4.15.1 | 0.000001 |
- |
pGlu-Trp-Pro-Arg-Pro-Gln-Ile-Pro-Pro |
pH 6.8, 25°C, reaction with (7-methoxycoumarin-2-acetic acid)-Ala-Ser-Asp-Lys-(N3-(2,4-dinitrophenyl)-L-2,3-diaminopropyl), C-domain |
650159 |
3.4.15.1 | 0.000001 |
- |
pGlu-Trp-Pro-Arg-Pro-Gln-Ile-Pro-Pro |
pH 6.8, 25°C, reaction with (7-methoxycoumarin-2-acetic acid)-Ser-Asp-Lys-(N3-(2,4-dinitrophenyl)-L-2,3-diaminopropyl), C-domain |
650159 |