EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.1.1.56 | -999 |
- |
Diethyl p-nitrophenyl phosphate |
double mutant W197I/C60H, spontaneous dephosphorylation below 1%, 22°C |
691005 |
3.1.1.56 | -999 |
- |
Diethyl p-nitrophenyl phosphate |
double mutant W197I/C60K, spontaneous dephosphorylation below 2%, 22°C |
691005 |
3.1.1.56 | -999 |
- |
Diethyl p-nitrophenyl phosphate |
double mutant W197I/C60Q, spontaneous dephosphorylation below 5%, 22°C |
691005 |
3.1.1.56 | -999 |
- |
Diethyl p-nitrophenyl phosphate |
double mutant W197I/C60R, spontaneous dephosphorylation below 1%, 22°C |
691005 |
3.1.1.56 | -999 |
- |
Diethyl p-nitrophenyl phosphate |
half maximal phosphorylation at inhibitor concentration of 0.38 +/-0.05 mM, mutant W197H, 22°C |
691005 |
3.1.1.56 | -999 |
- |
Diethyl p-nitrophenyl phosphate |
half maximal phosphorylation at inhibitor concentration of 0.6 +/-0.2 mM, double mutant W197I/C60K, 22°C |
691005 |
3.1.1.56 | -999 |
- |
Diethyl p-nitrophenyl phosphate |
half maximal phosphorylation at inhibitor concentration of 0.7 +/-0.1 mM, mutant W197I, 22°C |
691005 |
3.1.1.56 | -999 |
- |
Diethyl p-nitrophenyl phosphate |
half maximal phosphorylation at inhibitor concentration of 0.8 +/-0.6 mM, double mutant W197I/C60H, 22°C |
691005 |
3.1.1.56 | -999 |
- |
Diethyl p-nitrophenyl phosphate |
half maximal phosphorylation at inhibitor concentration of 1.04 +/-0.09 mM, double mutant W197I/C60R, 22°C |
691005 |
3.1.1.56 | -999 |
- |
Diethyl p-nitrophenyl phosphate |
half maximal phosphorylation at inhibitor concentration of 1.1 +/-0.3 mM, double mutant W197I/C60Q, 22°C |
691005 |