EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
2.7.1.105 | 0.095 |
- |
2,5-anhydro-D-mannitol 6-phosphate |
pH 7.5, 30°C |
640297 |
2.7.1.105 | 0.025 |
- |
3-(3-pyridinyl)-1-(4-pyridinyl)-2-propen-1-one |
inhibition of recombinant PFKFB3 protein, no inhibition of purified PFK-1 activity |
694113 |
2.7.1.105 | 0.16 |
- |
ADP |
pH 6.6, 25°C |
640284 |
2.7.1.105 | 0.008 |
- |
ATP |
pH 8.2, 30°C, mutant strain DF905 |
640323 |
2.7.1.105 | 0.01 |
- |
ATP |
pH 8.2, 30°C, mutant strain DF903 |
640323 |
2.7.1.105 | 8.5 |
- |
beta-D-fructose 6-phosphate |
pH 7.5, 30°C, recombinant HBP1 mutant S460D/T470D |
660814 |
2.7.1.105 | 9.2 |
- |
beta-D-fructose 6-phosphate |
pH 7.5, 30°C, recombinant HBP1 mutant S460D |
660814 |
2.7.1.105 | 9.5 |
- |
beta-D-fructose 6-phosphate |
pH 7.5, 30°C, recombinant HBP1 mutant H253A/S460D |
660814 |
2.7.1.105 | 9.6 |
- |
beta-D-fructose 6-phosphate |
pH 7.5, 30°C, recombinant His-tagged HBP1 deletion mutant |
660814 |
2.7.1.105 | 9.7 |
- |
beta-D-fructose 6-phosphate |
pH 7.5, 30°C, recombinant HBP1 mutant S477D |
660814 |