EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
2.5.1.78 | 0.0000008 |
- |
3-(1,3,7-trihydro-9-D-ribityl-2,6,8-purinetrione-7-yl)pentane 1-phosphate |
pH 7.0, 27°C |
688576 |
2.5.1.78 | 0.0000009 |
- |
3-(1,3,7-trihydro-9-D-ribityl-2,6,8-purinetrione-7-yl)pentane 1-phosphate |
pH 7.0, 27°C |
688576 |
2.5.1.78 | 0.0000013 |
- |
4-[4,6-dioxo-4,5,6,7-tetrahydro1-D-ribityl-1H-pyrazolo[3,4-d]-pyrimidin-3-yl]butyl 1-phosphate |
pH 7.0, 27°C |
688576 |
2.5.1.78 | 0.000002 |
- |
3-(1,3,7-trihydro-9-D-ribityl-2,6,8-purinetrione-7-yl)butane 1-phosphate |
pH 7.0, 27°C |
688576 |
2.5.1.78 | 0.0000037 |
- |
3-[4,6-dioxo-4,5,6,7-tetrahydro-1-D-ribityl-1H-pyrazolo[3,4-d]pyrimidin-3-yl]propyl 1-phosphate |
pH 7.0, 27°C |
688576 |
2.5.1.78 | 0.0000041 |
- |
1-deoxy-1-[2,6,8-trioxo-7-[4-(phosphonooxy)butyl]-1,2,3,6,7,8-hexahydro-9H-purin-9-yl]-D-ribitol |
pH 7.0, 37°C |
699719 |
2.5.1.78 | 0.0000041 |
- |
4-[4,6-dioxo-4,5,6,7-tetrahydro1-D-ribityl-1H-pyrazolo[3,4-d]-pyrimidin-3-yl]butyl 1-phosphate |
pH 7.0, 27°C |
688576 |
2.5.1.78 | 0.0000047 |
- |
1-deoxy-1-[2,6,8-trioxo-7-[5-(phosphonooxy)pentyl]-1,2,3,6,7,8-hexahydro-9H-purin-9-yl]-D-ribitol |
pH 7.0, 37°C |
699719 |
2.5.1.78 | 0.0000047 |
- |
5-[4,6-dioxo-4,5,6,7-tetrahydro-1-D-ribityl-1H-pyrazolo[3,4-d]pyrimidin-3-yl]pentyl 1-phosphate |
pH 7.0, 27°C |
688576 |
2.5.1.78 | 0.0000077 |
- |
5-[4,6-dioxo-4,5,6,7-tetrahydro-1-D-ribityl-1H-pyrazolo[3,4-d]pyrimidin-3-yl]pentyl 1-phosphate |
pH 7.0, 27°C |
688576 |