EC Number   |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor  |
Reference |
|---|
    1.3.1.22 | 0.000006 |
- |
(+)-LY191704 |
- |
656656 |
| 1.3.1.22 | 0.000004 |
- |
(-)-LY191704 |
- |
656656 |
| 1.3.1.22 | 0.00092 |
- |
(10bR)-8-chloro-4,10b-dimethyl-4a,5,6,10b-tetrahydrophenanthridin-2(1H)-one |
isoform I |
656656 |
| 1.3.1.22 | 0.0011 |
- |
(10bR)-8-chloro-4,5,10b-trimethyl-4a,5,6,10b-tetrahydrophenanthridin-2(1H)-one |
isoform I |
656656 |
| 1.3.1.22 | 0.00026 |
- |
(4aS)-7-chloro-4a-methyl-2,3,4,4a-tetrahydrophenanthrene-2-carboxylic acid |
isoform II, Ki,app-value |
656656 |
| 1.3.1.22 | 0.0012 |
- |
(4aS)-7-chloro-4a-methyl-2,3,4,4a-tetrahydrophenanthrene-2-carboxylic acid |
isoform I, Ki,app-value |
656656 |
| 1.3.1.22 | 0.000035 |
- |
(5alpha,20-R)-4-Diazo-21-hydroxy-20-methylpregnan-3-one |
at 25°C formation of the reversible EI complex is not rate-limiting for enzyme inactivation, and this is expressed as saturation kinetics for the inhibition reaction |
396204 |
| 1.3.1.22 | 0.000085 |
- |
17-diisopropylcarbamoyl-2-androsten-3-carboxylate |
- |
390657 |
| 1.3.1.22 | 0.000007 |
0.000018 |
17-diisopropylcarbamoyl-3,5-androstadien-3-carboxylate |
- |
390657 |
| 1.3.1.22 | 0.00003 |
- |
17-diisopropylcarbamoyl-3-androsten-3-carboxyate |
- |
390657 |
