EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
1.1.1.43 | 0.002 |
- |
metochloropramide |
25°C, pH 8.0, non-competitive inhibition |
712601 |
1.1.1.43 | 0.0042 |
- |
5-(3alpha,7alpha,12alpha-triacetoxy-5-beta-cholanamido)-1,3,4-thiadiazole-2-sulfonamide |
- |
688050 |
1.1.1.43 | 0.006 |
- |
4-[(1R,2S)-1-hydroxy-2-{[2-(4-hydroxyphenyl)ethyl]amino}propyl]phenol |
25°C, pH 8.0, non-competitive inhibition |
712601 |
1.1.1.43 | 0.008 |
- |
ketotifen |
25°C, pH 8.0, non-competitive inhibition |
712601 |
1.1.1.43 | 0.01 |
- |
dacarbazine |
25°C, pH 8.0, non-competitive inhibition |
712601 |
1.1.1.43 | 0.05 |
- |
meloxicam |
25°C, pH 8.0, non-competitive inhibition |
712601 |
1.1.1.43 | 0.0734 |
- |
gadopentetic acid |
25°C, pH 8.0, non-competitive inhibition |
712601 |
1.1.1.43 | 0.0878 |
- |
5-(3alpha,7alpha,12alpha-trihydroxy-5-beta-cholanamido)-1,3,4-thiadiazole-2-sulfonamide |
- |
688050 |
1.1.1.43 | 0.127 |
- |
Furosemide |
25°C, pH 8.0, non-competitive inhibition |
712601 |
1.1.1.43 | 0.136 |
- |
methotrexate |
25°C, pH 8.0, non-competitive inhibition |
712601 |