EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
1.1.1.153 | 0.0002 |
- |
N-acetyl-serotonin |
pH 6.4, 25°C, brain enzyme |
286023 |
1.1.1.153 | 0.03 |
- |
Melatonin |
pH 6.4, 25°C, brain enzyme |
286023 |
1.1.1.153 | 2.3 |
- |
serotonin |
pH 6.4, 25°C, brain enzyme |
286023 |
1.1.1.153 | 3.4 |
- |
1-norepinephrine |
pH 6.4, 25°C, brain enzyme |
286023 |
1.1.1.153 | 0.00017 |
- |
N-acetyl-serotonin |
pH 6.4, 25°C, erythrocyte enzyme |
286023 |
1.1.1.153 | 0.025 |
- |
Melatonin |
pH 6.4, 25°C, erythrocyte enzyme |
286023 |
1.1.1.153 | 2.5 |
- |
serotonin |
pH 6.4, 25°C, erythrocyte enzyme |
286023 |
1.1.1.153 | 3.1 |
- |
1-norepinephrine |
pH 6.4, 25°C, erythrocyte enzyme |
286023 |
1.1.1.153 | 0.0005 |
- |
phenylquinone |
wild-type, pH 6.7, 37°C |
725527 |
1.1.1.153 | 0.0009 |
- |
benzoquinone |
wild-type, pH 6.7, 37°C |
725527 |