EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
4.3.1.B2 | 0.00067 |
- |
N1-[(5'-phosphoarabinitolyl)-formimino]-5-aminoimidazole-4-carboxamide ribonucleotide |
pH 7.0, 30°C, substrate: N1-[(5'-phosphoribulosyl)formimino]-5-aminoimidazole-4-carboxamido-1-beta-D-ribofuranosyl 5'-phosphate |
726939 |
4.3.1.B2 | 0.0016 |
- |
N1-[(5'-phosphoarabinitolyl)-formimino]-5-aminoimidazole-4-carboxamide ribonucleotide |
pH 7.0, 30°C, substrate: L-glutamine, uncompetitive inhibition constant |
726939 |
4.3.1.B2 | 0.003 |
- |
N1-[(5'-phosphoarabinitolyl)-formimino]-5-aminoimidazole-4-carboxamide ribonucleotide |
pH 7.0, 30°C, substrate: L-glutamine, competitive inhibition constant |
726939 |
4.3.1.B2 | 0.004 |
- |
N1-[(5'-phosphoribitolyl)-formimino]-5-aminoimidazole-4-carboxamide ribonucleotide |
pH 7.0, 30°C, N1-[(5'-phosphoribulosyl)formimino]-5-aminoimidazole-4-carboxamido-1-beta-D-ribofuranosyl 5'-phosphate |
726939 |
4.3.1.B2 | 0.38 |
- |
albizziin |
pH 7.0, 30°C, substrate: L-glutamine |
726939 |
4.3.1.B2 | 0.6 |
- |
albizziin |
pH 7.0, 30°C, competitive inhibition constant, substrate: N1-[(5'-phosphoribulosyl)formimino]-5-aminoimidazole-4-carboxamido-1-beta-D-ribofuranosyl 5'-phosphate |
726939 |
4.3.1.B2 | 1.6 |
- |
albizziin |
pH 7.0, 30°C, uncompetitive inhibition constant, substrate: N1-[(5'-phosphoribulosyl)formimino]-5-aminoimidazole-4-carboxamido-1-beta-D-ribofuranosyl 5'-phosphate |
726939 |