EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.5.3.1 | 0.0009 |
- |
2-(S)-amino-6-boronohexanoic acid |
pH 8.0, 21°C |
752398 |
3.5.3.1 | 0.0011 |
- |
(DL)-2-amino-6-borono-2-[1-(3,4-dichlorobenzyl)piperidin-4-yl]-hexanoic acid |
pH 8.0, 21°C |
752398 |
3.5.3.1 | 0.0014 |
- |
(S)-2-amino-6-borono-2-[2-(piperidin-1-yl)ethyl]hexanoic acid |
pH 8.0, 21°C |
752398 |
3.5.3.1 | 0.0016 |
- |
Nomega-hydroxy-L-arginine |
pH 7.5, 22°C |
654612 |
3.5.3.1 | 0.0036 |
- |
S-(2-boronoethyl)-L-cysteine |
pH 9.5, 25°C, supramolecular tandem assay method |
704175 |
3.5.3.1 | 0.004 |
- |
2-(S)-amino-5-(2-aminoimidazol-1-yl)pentanoic acid |
pH not specified in the publication, temperature not specified in the publication |
712701 |
3.5.3.1 | 0.0045 |
- |
S-(2-boronoethyl)-L-cysteine |
T135A mutant |
696307 |
3.5.3.1 | 0.01 |
- |
2(S)-amino-6-boronohexanoic acid |
mutant dN-PFA, pH 8.5, 37°C |
711253 |
3.5.3.1 | 0.011 |
- |
2(S)-amino-6-boronohexanoic acid |
mutant dN-PFA, pH 7.4, 37°C |
711253 |
3.5.3.1 | 0.012 |
- |
2(S)-amino-6-boronohexanoic acid |
mutant dN-PFA, pH 8.0, 37°C |
711253 |