EC Number   |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
|---|
   3.4.22.69 | 0.0452 |
- |
N-[(benzyloxy)carbonyl]-L-valyl-N-[(2S)-1,5-dioxo-1,5-di(1,3-thiazol-2-yl)pentan-2-yl]-L-leucinamide |
- |
707665 |
| 3.4.22.69 | 0.0493 |
- |
benzyl [(2S)-1-[[(2S)-1-[[(2S)-1-(1,3-benzothiazol-2-yl)-5-(diethylamino)-1,5-dioxopentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]carbamate |
- |
707665 |
| 3.4.22.69 | 0.052 |
- |
benzyl ((S)-1-(((S)-1-(5-(4-methoxyphenyl)thiazol-2-yl)-1-oxo-3-((S)-2-oxopyrrolidin-3-yl)propan-2-yl)amino)-4-methyl-1-oxopentan-2-yl)carbamate |
enzyme mutant R188I, pH and temperature not specified in the publication |
731748 |
| 3.4.22.69 | 0.061 |
- |
1-[bis(4-chlorophenyl)methyl]-3-[2-[(2,4-dichlorobenzyl)oxy]-2-(2,4-dichlorophenyl)ethyl]-1H-imidazol-3-ium |
- |
679402 |
| 3.4.22.69 | 0.07273 |
- |
N-acetyl-NSTSQ |
in 40 mM Tris-HCl buffer, pH 7.3, temperature not specified in the publication |
717101 |
| 3.4.22.69 | 0.112 |
- |
benzyl [(2S)-1-[[(2S)-1-[[(2S)-5-(diethylamino)-1,5-dioxo-1-(1,3-thiazol-2-yl)pentan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]carbamate |
- |
707665 |
| 3.4.22.69 | 0.116 |
- |
N-[(benzyloxy)carbonyl]-L-valyl-N-[(3S)-5-carboxy-1,1,1-trifluoro-2-oxopentan-3-yl]-L-leucinamide |
- |
707665 |
| 3.4.22.69 | 0.126 |
- |
Val-Thr-Phe-Gln |
pH 7.5, 30°C |
755253 |
| 3.4.22.69 | 0.135 |
- |
N-[(benzyloxy)carbonyl]-L-alanyl-L-valyl-N-[(3S)-6-amino-1,1,1-trifluoro-2,6-dioxohexan-3-yl]-L-leucinamide |
- |
707665 |
| 3.4.22.69 | 0.159 |
- |
benzyl [(2S)-1-[[(2S)-1-(1,3-benzothiazol-2-yl)-5-(diethylamino)-1,5-dioxopentan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]carbamate |
- |
707665 |
