EC Number |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
---|
3.4.22.62 | 0.0008 |
- |
Zn2+ |
mutant C287A, pH 6.5, 37°C |
732880 |
3.4.22.62 | 0.0008 |
- |
Zn2+ |
mutant H237A, pH 6.5, 37°C |
732880 |
3.4.22.62 | 0.00097 |
- |
acetyl-YVAD-CHO |
pH 7.5, 25°C |
647423 |
3.4.22.62 | 0.0012 |
- |
Zn2+ |
mutant C239S, pH 6.5, 37°C |
732880 |
3.4.22.62 | 0.0015 |
- |
Zn2+ |
mutant C172A, pH 6.5, 37°C |
732880 |
3.4.22.62 | 0.0018 |
- |
Zn2+ |
wild-type enzyme, pH 6.5, 37°C |
732880 |
3.4.22.62 | 0.00233 |
- |
(3S,6S,8aS)-6-(L-alanylamino)-N-(diphenylmethyl)-5-oxooctahydroindolizine-3-carboxamide |
pH and temperature not specified in the publication |
731452 |
3.4.22.62 | 0.0142 |
- |
benzyloxycarbonyl-VAE-fluoromethylketone |
- |
666835 |
3.4.22.62 | 0.0171 |
- |
benzyloxycarbonyl-VAD-fluoromethylketone |
- |
666835 |