EC Number   |
Ki Value [mM] |
Ki Value maximum [mM] |
Inhibitor |
Reference |
|---|
   3.4.21.27 | 0.00253 |
- |
trans-4-(aminomethyl)-N-[1-(1-oxido-2-phenylpyridin-4-yl)-2-phenylethyl]cyclohexanecarboxamide |
pH and temperature not specified in the publication |
731466 |
| 3.4.21.27 | 0.00286 |
- |
4-(2-((S)-1-(trans-4-(aminomethyl)cyclohexanecarboxamido)-2-phenylethyl)-1H-imidazol-4-yl)-N,N-dimethylbenzamide |
at pH 7.4 and 37°C |
732318 |
| 3.4.21.27 | 0.0029 |
- |
trans-N-[(1S)-1-[4-(3-amino-1H-indazol-6-yl)-5-chloro-1H-imidazol-2-yl]-2-phenylethyl]cyclohexane-1,4-dicarboxamide |
at 25°C, pH not specified in the publication |
731462 |
| 3.4.21.27 | 0.003074 |
- |
trans-4-(aminomethyl)-N-((S)-1-(5-oxo-1-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)-2-phenylethyl)cyclohexanecarboxamide |
at pH 7.4 and 37°C |
732318 |
| 3.4.21.27 | 0.0064 |
- |
methyl [(9S)-9-([(2E)-3-[5-chloro-2-(1H-tetrazol-1-yl)phenyl]prop-2-enoyl]amino)-3-oxo-1,2,3,8,9,11-hexahydro-13,10-(azeno)-4,7-etheno-2,11-benzodiazacyclopentadecin-16-yl]carbamate |
at 25°C, pH not specified in the publication |
752995 |
| 3.4.21.27 | 0.00694 |
- |
trans-4-(aminomethyl)-N-((S)-2-phenyl-1-(3-phenyl-1H-pyrazol-5-yl)ethyl)cyclohexanecarboxamide |
at pH 7.4 and 37°C |
732318 |
| 3.4.21.27 | 0.0081 |
- |
methyl [(9S)-12-chloro-9-([(2E)-3-[5-chloro-2-(1H-tetrazol-1-yl)phenyl]prop-2-enoyl]amino)-3-oxo-1,2,3,8,9,11-hexahydro-13,10-(azeno)-4,7-etheno-2,11-benzodiazacyclopentadecin-16-yl]carbamate |
at 25°C, pH not specified in the publication |
752995 |
| 3.4.21.27 | 0.01142 |
- |
trans-4-(aminomethyl)-N-[2-phenyl-1-(4-phenylpyrimidin-2-yl)ethyl]cyclohexanecarboxamide |
pH and temperature not specified in the publication |
731466 |
| 3.4.21.27 | 0.03021 |
- |
trans-4-(aminomethyl)-N-[2-phenyl-1-(6-phenylpyridin-2-yl)ethyl]cyclohexanecarboxamide |
pH and temperature not specified in the publication |
731466 |
| 3.4.21.27 | 0.06 |
- |
4-aminobenzamidine |
37°C, recombinant wild-type enzyme, versus substrate S-2366 |
683167 |
