EC Number |
KM Value [mM] |
KM Value Maximum [mM] |
Substrate |
Reference |
---|
3.4.22.48 | 0.0056 |
- |
2-aminobenzoyl-Phe-Gly-Ala-Lys-5-amino-2-nitrobenzoylamide |
pH 7.6, 37°C, staphopain A |
717294 |
3.4.22.48 | 0.0076 |
- |
2-aminobenzoyl-Ile-Ala-Ala-Gly-5-amino-2-nitrobenzoylamide |
pH 7.6, 37°C, staphopain A |
717294 |
3.4.22.48 | 0.014 |
- |
2-aminobenzoyl-Ile-Ala-Lys-Asp-5-amino-2-nitrobenzoylamide |
pH 7.6, 37°C, staphopain C |
717294 |
3.4.22.48 | 0.032 |
- |
cystatin D |
Ala10 bond hydrolyzed by staphopain A, truncation of cystatin D shown to cause alleviated inhibition of endogenous target enzymes investigated, disturbance of the host protease-inhibitor balance |
683205 |
3.4.22.48 | 0.033 |
- |
cystatin C |
Gly11 bond hydrolyzed by staphopain A, N-terminal truncation shown to impair inhibition of additional targets, disturbance of the host protease-inhibitor balance |
683205 |
3.4.22.48 | 0.154 |
- |
2-aminobenzoyl-Phe-Gly-Ala-Lys-5-amino-2-nitrobenzoylamide |
pH 7.6, 37°C, staphopain A |
717294 |
3.4.22.48 | 0.1639 |
- |
2-aminobenzoyl-Ile-Ala-Ala-Gly-5-amino-2-nitrobenzoylamide |
pH 7.6, 37°C, staphopain A |
717294 |
3.4.22.48 | 0.271 |
- |
2-aminobenzoyl-Ile-Ala-Ala-Gly-5-amino-2-nitrobenzoylamide |
pH 7.6, 37°C, staphopain C |
717294 |
3.4.22.48 | 0.385 |
- |
2-aminobenzoyl-Phe-Gly-Ala-Lys-5-amino-2-nitrobenzoylamide |
pH 7.6, 37°C, staphopain C |
717294 |
3.4.22.48 | 0.5 |
- |
N-benzyloxycarbonyl-Phe-Leu-Glu-NH-p-nitroanilide |
pH 8.0-8.8 |
643963 |