EC Number |
Inhibitors |
Structure |
---|
3.4.99.B2 | 1,10-phenanthroline |
0.1 mM, 8.3% inhibition |
|
3.4.99.B2 | Aprotinin |
0.1 mM, 14% inhibition |
|
3.4.99.B2 | benzoyl-Arg-His-D-Asp-CH2Cl |
1 mM, about 70% inhibition of paenidase I and II |
|
3.4.99.B2 | benzoyl-Arg-His-[D-Asp]-CH2Cl |
0.1 mM, 48% residual activity |
|
3.4.99.B2 | benzoyl-L-Arg-L-His-D-Asp-CH2Cl |
0.003 mM, 50% inhibition |
|
3.4.99.B2 | biotinyl-(epsilon-aminocaproic acid)-L-Arg-L-His-D-Asp-CH2Cl |
- |
|
3.4.99.B2 | Co2+ |
1.0 mM, 31% inhibition of paenidase I, 46% inhibition of paenidase II |
|
3.4.99.B2 | diisopropyl fluorophosphate |
at 0.5 mM, 15.5% inhibition |
|
3.4.99.B2 | lactacystin |
- |
|
3.4.99.B2 | leupeptin |
0.03 mM, 8.5% inhibition |
|