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Results 1 - 10 of 89 > >>
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EC Number Inhibitors Commentary Structure
Display the reaction diagram Show all sequences 3.4.21.1221-[(2R)-4-(4-benzylpiperazin-1-yl)-4-oxo-2-[(phenylmethanesulfonyl)amino]butanoyl]-N-[(4-carbamimidoylphenyl)methyl]-L-prolinamide - Go to the Ligand Summary Page
Display the reaction diagram Show all sequences 3.4.21.1223-cyclohexyl-N-(phenylmethanesulfonyl)-D-alanyl-N-[(4-carbamimidoylphenyl)methyl]-N6-decanoyl-L-lysinamide peptide mimetic inhibitor. Cleavage of HA0 and the spread of A/Hamburg/09 in TMPRSS2-expressing cells are strongly inhibited by the decanoylated inhibitor. Only low amounts of progeny virions are detected in supernatants of inhibitor-treated cells at 24 h p.i. due to the suppression of proteolytic activation of HA and thus the suppression of virus propagation Go to the Ligand Summary Page
Display the reaction diagram Show all sequences 3.4.21.1223-[(2S)-2-[(2',4'-dichloro[1,1'-biphenyl]-3-sulfonyl)amino]-3-(4-[2-[(methylcarbamoyl)amino]ethyl]piperidin-1-yl)-3-oxopropyl]benzene-1-carboximidamide - Go to the Ligand Summary Page
Display the reaction diagram Show all sequences 3.4.21.1223-[(2S)-2-[(2',4'-dimethoxy[1,1'-biphenyl]-3-sulfonyl)amino]-3-(4-[2-[(methylcarbamoyl)amino]ethyl]piperidin-1-yl)-3-oxopropyl]benzene-1-carboximidamide - Go to the Ligand Summary Page
Display the reaction diagram Show all sequences 3.4.21.1223-[(2S)-3-[4-(2-aminoethyl)piperidin-1-yl]-2-[(2',4'-dichloro[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide treatment of cells with 10 microM inhibitor causes a 10fold and 100fold reduction in virus titres of A/Hamburg H1N1 and A/Aichi H3N2 respectively, at 24 h Go to the Ligand Summary Page
Display the reaction diagram Show all sequences 3.4.21.1223-[(2S)-3-[4-[(cyclohexylcarbamoyl)amino]piperidin-1-yl]-2-[(2',4'-dichloro[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide - Go to the Ligand Summary Page
Display the reaction diagram Show all sequences 3.4.21.1223-[(2S)-3-[4-[(cyclohexylcarbamoyl)amino]piperidin-1-yl]-2-[(2',4'-dimethoxy[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide - Go to the Ligand Summary Page
Display the reaction diagram Show all sequences 3.4.21.1223-[(2S)-3-[4-[2-([[4-(2-aminoethyl)cyclohexyl]carbamoyl]amino)ethyl]piperidin-1-yl]-2-[(2',3'-dichloro[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide - Go to the Ligand Summary Page
Display the reaction diagram Show all sequences 3.4.21.1223-[(2S)-3-[4-[2-([[4-(2-aminoethyl)cyclohexyl]carbamoyl]amino)ethyl]piperidin-1-yl]-2-[(2',4'-dichloro[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide - Go to the Ligand Summary Page
Display the reaction diagram Show all sequences 3.4.21.1223-[(2S)-3-[4-[2-([[4-(2-aminoethyl)cyclohexyl]carbamoyl]amino)ethyl]piperidin-1-yl]-2-[(2',4'-dimethoxy[1,1'-biphenyl]-3-sulfonyl)amino]-3-oxopropyl]benzene-1-carboximidamide - Go to the Ligand Summary Page
Results 1 - 10 of 89 > >>
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