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Results 1 - 10 of 70 > >>
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EC Number Inhibitors Commentary Structure
Display the word mapDisplay the reaction diagram Show all sequences 3.4.21.112(2R,2'R)-2,2'-[(E)-diazene-1,2-diylbis[benzene-2,1-diyloxy(1-oxoethane-2,1-diyl)imino[(2S)-1-oxo-4-phenylbutane-2,1-diyl]imino]]bis(3-phenylpropanoic acid) - Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 3.4.21.112(2S,2'S)-2,2'-[(E)-diazene-1,2-diylbis[benzene-2,1-diyloxy(1-oxoethane-2,1-diyl)imino]]bis(3-methylbutanoic acid) - Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 3.4.21.112(2S,2'S)-2,2'-[(E)-diazene-1,2-diylbis[benzene-2,1-diyloxy(1-oxoethane-2,1-diyl)imino]]bis(4-phenylbutanoic acid) - Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 3.4.21.112(3S,4S,5S,6R)-2-([(2R,3S,4S,5S,6S)-3,5-dihydroxy-2-(hydroxymethyl)-6-methoxytetrahydro-2H-pyran-4-yl]amino)-6-(hydroxymethyl)tetrahydro-2H-thiopyran-3,4,5-triol i.e. BJ-12-26-1, greatly reduces SKI-1 zymogen processing, and abolishes the processing of substrate SREBP-2 Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 3.4.21.112(3S,4S,5S,6R)-2-([(2S,3S,4R,5S,6R)-4,5-dihydroxy-6-(hydroxymethyl)-2-methoxytetrahydro-2H-pyran-3-yl]amino)-6-(hydroxymethyl)tetrahydro-2H-thiopyran-3,4,5-triol i.e. BJ-12-21-2, greatly reduces SKI-1 zymogen processing, and abolishes the processing of substrate SREBP-2 Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 3.4.21.112(R)-4-((diethylamino)methyl)-N-(2-methoxyphenethyl)-N-(pyrrolidin-3-yl)benzamide inhibits endogenous SREBP processing in Chinese hamster ovary cells. Compound down-regulates the signal from an SRE-luciferase reporter gene in human embryonic kidney 293 cells and the expression of endogenous SREBP target genes in cultured HepG2 cells. In mice treated with the compound for 24 h, the expression of hepatic SREBP target genes is suppressed, and the hepatic rates of cholesterol and fatty acid synthesis are reduced Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 3.4.21.112(S)-4-((diethylamino)methyl)-N-(2-methoxyphenethyl)-N-(pyrrolidin-3-yl)benzamide purified S-enantiomer Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 3.4.21.1121,10-phenanthroline partial inhibition at very high concentrations Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 3.4.21.1121,10-phenanthroline complete inactivation at 5 mM Go to the Ligand Summary Page
Display the word mapDisplay the reaction diagram Show all sequences 3.4.21.1121-(4-[[2-(2-methoxyphenyl)ethyl](pyrrolidin-3-yl)carbamoyl]benzyl)piperidine-3-carboxamide - Go to the Ligand Summary Page
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