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Literature summary extracted from

  • Brandstetter, H.; Turk, D.; Hoeffken, H.W.; Grosse, D.; Sturzebecher, J.; Martin, P.D.; Edwards, B.F.; Bode, W.
    Refined 2.3 A X-ray crystal structure of bovine thrombin complexes formed with the benzamidine and arginine-based thrombin inhibitors NAPAP, 4-TAPAP and MQPA. A starting point for improving antithrombotics (1992), J. Mol. Biol., 226, 1085-1099.
    View publication on PubMed

Crystallization (Commentary)

EC Number Crystallization (Comment) Organism
3.4.21.5 enzyme complex formed with the benzamidine and Arg-based thrombin inhibitors Nalpha-(2-naphthalenesulfonyl)-glycyl-D-3-aminophenyl-alanyl-piperidine, N-alpha-tosyl-(3-amidinophenyl)alanine piperidine and (2R,4R)-4-methyl-1-[Nalpha-(3-methyl-1,2,3,4-tetrahydro-8-quinolinesulfonyl)-L-arginyl]-2-piperidine carboxylic acid Bos taurus

Organism

EC Number Organism UniProt Comment Textmining
3.4.21.5 Bos taurus
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