EC Number | Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|---|
7.6.2.2 | plasma membrane | - |
Homo sapiens | 5886 | - |
EC Number | Organism | UniProt | Comment | Textmining |
---|---|---|---|---|
7.6.2.2 | Homo sapiens | Q2M3G0 | - |
- |
7.6.2.2 | Homo sapiens | Q8HXQ5 | - |
- |
7.6.2.2 | Homo sapiens | Q9UNQ0 | - |
- |
EC Number | Source Tissue | Comment | Organism | Textmining |
---|---|---|---|---|
7.6.2.2 | enterocyte | BCRP | Homo sapiens | - |
7.6.2.2 | hepatocyte | - |
Homo sapiens | - |
EC Number | Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|---|
7.6.2.2 | ATP + H2O + acridine orange[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + acridine orange[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + aflatoxin B[side 1] | substrate for MRP1 | Homo sapiens | ADP + phosphate + aflatoxin B[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + amiodarone[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + amiodarone[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + arsenite[side 1] | substrate for MRP1 | Homo sapiens | ADP + phosphate + arsenite[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + azidopine[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + azidopine[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + bilirubin[side 1] | substrate for MRP1 | Homo sapiens | ADP + phosphate + bilirubin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + calcein[side 1] | substrate for MRP1 | Homo sapiens | ADP + phosphate + calcein[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + calphostin C[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + calphostin C[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + clorambucil[side 1] | substrate for MRP1 | Homo sapiens | ADP + phosphate + clorambucil[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + colchicine[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + colchicine[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + cyclophosphamide[side 1] | substrate for MRP1 | Homo sapiens | ADP + phosphate + cyclophosphamide[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + cyclosporine[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + cyclosporine[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + daunorubicin[side 1] | substrate for BCRP | Homo sapiens | ADP + phosphate + daunorubicin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + daunorubicin[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + daunorubicin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + dehydroepiandrosterone sulfate[side 1] | substrate for MRP1 | Homo sapiens | ADP + phosphate + dehydroepiandrosterone sulfate[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + dinitrophenyl[side 1] | substrate for MRP1 | Homo sapiens | ADP + phosphate + dinitrophenyl[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + dipyridamole[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + dipyridamole[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + doxorubicin[side 1] | substrate for P-glycoprotein, BCRP, and MRP1 | Homo sapiens | ADP + phosphate + doxorubicin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + erythromycin[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + erythromycin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + estradiol[side 1] | substrate for MRP1 | Homo sapiens | ADP + phosphate + estradiol[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + estrone-3-sulfate[side 1] | substrate for BCRP | Homo sapiens | ADP + phosphate + estrone-3-sulfate[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + estrone[side 1] | substrate for MRP1 | Homo sapiens | ADP + phosphate + estrone[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + ethacrynic acid[side 1] | substrate for MRP1 | Homo sapiens | ADP + phosphate + ethacrynic acid[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + etoposide[side 1] | substrate for MRP1 | Homo sapiens | ADP + phosphate + etoposide[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + FK-506[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + FK-506[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + folic acid[side 1] | substrate for MRP1 | Homo sapiens | ADP + phosphate + folic acid[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + gefitinib[side 1] | substrate for BCRP | Homo sapiens | ADP + phosphate + gefitinib[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + genistein[side 1] | substrate for BCRP | Homo sapiens | ADP + phosphate + genistein[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + genistein[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + genistein[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + glutathione disulfide[side 1] | substrate for MRP1 | Homo sapiens | ADP + phosphate + glutathione disulfide[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + hematoporphyrin[side 1] | substrate for BCRP | Homo sapiens | ADP + phosphate + hematoporphyrin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + indinavir[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + indinavir[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + leucovorin[side 1] | substrate for MRP1 | Homo sapiens | ADP + phosphate + leucovorin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + leukotriene C4[side 1] | substrate for MRP1 | Homo sapiens | ADP + phosphate + leukotriene C4[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + leukotriene D4[side 1] | substrate for MRP1 | Homo sapiens | ADP + phosphate + leukotriene D4[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + melphalan[side 1] | substrate for MRP1 | Homo sapiens | ADP + phosphate + melphalan[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + methotrexate[side 1] | substrate for BCRP | Homo sapiens | ADP + phosphate + methotrexate[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + mitomycin C[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + mitomycin C[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + mitoxantrone[side 1] | substrate for BCRP | Homo sapiens | ADP + phosphate + mitoxantrone[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + progesterone[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + progesterone[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + prostaglandin E2[side 1] | substrate for MRP1 | Homo sapiens | ADP + phosphate + prostaglandin E2[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + PSC-833[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + PSC-833[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + quercetin[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + quercetin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + quinidine[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + quinidine[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + rapamycin[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + rapamycin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + rhodamine 123[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + rhodamine 123[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + riboflavin[side 1] | substrate for BCRP | Homo sapiens | ADP + phosphate + riboflavin[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + ritonavir[side 1] | substrate for P-glycoprotein and MRP1 | Homo sapiens | ADP + phosphate + ritonavir[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + staurosporine[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + staurosporine[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + tamoxifen[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + tamoxifen[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + taxol[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + taxol[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + teniposide[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + teniposide[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + verapamil[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + verapamil[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + vinblastine[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + vinblastine[side 2] | - |
? | |
7.6.2.2 | ATP + H2O + vincristine[side 1] | substrate for P-glycoprotein | Homo sapiens | ADP + phosphate + vincristine[side 2] | - |
? |
EC Number | Synonyms | Comment | Organism |
---|---|---|---|
7.6.2.2 | ABCG2 | - |
Homo sapiens |
7.6.2.2 | BCRP | - |
Homo sapiens |
7.6.2.2 | breast cancer resistance protein | - |
Homo sapiens |
7.6.2.2 | canalicular multispecific organic anion transporter | - |
Homo sapiens |
7.6.2.2 | cMOAT | - |
Homo sapiens |
7.6.2.2 | MRP1 | - |
Homo sapiens |
7.6.2.2 | multidrugresistance 1 | - |
Homo sapiens |
7.6.2.2 | P-glycoprotein | - |
Homo sapiens |
7.6.2.2 | Pgp | - |
Homo sapiens |