EC Number | Activating Compound | Comment | Organism | Structure |
---|---|---|---|---|
2.3.2.5 | EDTA | the enzymatic activity increases by about 55% in the presence of 1 mM EDTA | Ixodes scapularis |
EC Number | Cloned (Comment) | Organism |
---|---|---|
2.3.2.5 | expressed in Escherichia coli BL21(DE3) CodonPlus-RIL cells | Ixodes scapularis |
EC Number | Crystallization (Comment) | Organism |
---|---|---|
2.3.2.5 | sitting drop vapor diffusion method, using 10% (w/v) PEG 8000, 8% (v/v) ethylene glycol, 0.1 M HEPES pH 7.5 | Ixodes scapularis |
EC Number | Inhibitors | Comment | Organism | Structure |
---|---|---|---|---|
2.3.2.5 | 1,10-phenanthroline | - |
Ixodes scapularis | |
2.3.2.5 | 1-Benzylimidazole | - |
Ixodes scapularis | |
2.3.2.5 | dipicolinic acid | - |
Ixodes scapularis | |
2.3.2.5 | Nomega-acetylhistamine | - |
Ixodes scapularis | |
2.3.2.5 | PBD150 | - |
Ixodes scapularis |
EC Number | KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|---|
2.3.2.5 | 0.0218 | - |
L-glutaminyl 2-naphthylamide | at pH 8.0 and 25°C | Ixodes scapularis |
EC Number | Metals/Ions | Comment | Organism | Structure |
---|---|---|---|---|
2.3.2.5 | additional information | the enzyme is metal-independent | Ixodes scapularis | |
2.3.2.5 | Zn2+ | 0.5 mol of zinc per mole of enzyme | Ixodes scapularis |
EC Number | Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|---|
2.3.2.5 | L-glutaminyl-peptide | Ixodes scapularis | - |
5-oxoprolyl-peptide + NH3 | - |
? |
EC Number | Organism | UniProt | Comment | Textmining |
---|---|---|---|---|
2.3.2.5 | Ixodes scapularis | B7QK46 | - |
- |
EC Number | Purification (Comment) | Organism |
---|---|---|
2.3.2.5 | Ni-NTA column chromatography and Sephacryl S-100 gel filtration | Ixodes scapularis |
EC Number | Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|---|
2.3.2.5 | L-glutaminyl 2-naphthylamide | - |
Ixodes scapularis | L-glutamine + 2-naphthylamine | - |
? | |
2.3.2.5 | L-glutaminyl-peptide | - |
Ixodes scapularis | 5-oxoprolyl-peptide + NH3 | - |
? |
EC Number | Synonyms | Comment | Organism |
---|---|---|---|
2.3.2.5 | glutaminyl cyclase | - |
Ixodes scapularis |
EC Number | Temperature Stability Minimum [°C] | Temperature Stability Maximum [°C] | Comment | Organism |
---|---|---|---|---|
2.3.2.5 | 53 | - |
melting temperature | Ixodes scapularis |
EC Number | Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|---|
2.3.2.5 | 8.8 | - |
L-glutaminyl 2-naphthylamide | at pH 8.0 and 25°C | Ixodes scapularis |
EC Number | Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|---|
2.3.2.5 | 0.000342 | - |
PBD150 | at pH 8.0 and 25°C | Ixodes scapularis | |
2.3.2.5 | 0.00345 | - |
1,10-phenanthroline | at pH 8.0 and 25°C | Ixodes scapularis | |
2.3.2.5 | 0.0102 | - |
1-Benzylimidazole | at pH 8.0 and 25°C | Ixodes scapularis | |
2.3.2.5 | 0.0142 | - |
Nomega-acetylhistamine | at pH 8.0 and 25°C | Ixodes scapularis | |
2.3.2.5 | 0.0368 | - |
dipicolinic acid | at pH 8.0 and 25°C | Ixodes scapularis |