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Literature summary extracted from

  • Sanchez-Fernandez, E.M.; Alvarez, E.; Ortiz Mellet, C.; Garcia Fernandez, J.M.
    Synthesis of multibranched australine derivatives from reducing castanospermine analogues through the amadori rearrangement of gem-diamine intermediates: selective inhibitors of beta-glucosidase (2014), J. Org. Chem., 79, 11722-11728.
    View publication on PubMed

Inhibitors

EC Number Inhibitors Comment Organism Structure
3.2.1.21 3,8-dibutylamino-7,8-dideoxy-5-octylimino-6-oxa-3-epi-australine
-
 Bos taurus
3.2.1.21 3,8-dibutylamino-7,8-dideoxy-5-octylimino-6-oxa-3-epi-australine
-
 Prunus dulcis
3.2.1.21 7,8-dideoxy-3,8-didodecylamino-5-octylimino-6-oxa-3-epi-australine
-
 Bos taurus
3.2.1.21 7,8-dideoxy-3,8-didodecylamino-5-octylimino-6-oxa-3-epi-australine
-
 Prunus dulcis
3.2.1.21 7,8-dideoxy-3,8-dioctylamino-5-octylimino-6-oxa-3-epi-australine
-
 Bos taurus
3.2.1.21 7,8-dideoxy-3,8-dioctylamino-5-octylimino-6-oxa-3-epi-australine
-
 Prunus dulcis
3.2.1.21 7,8-dideoxy-3-hydroxy-8-octylamino-5-octylimino-6-oxa-3-epi-australine
-
 Bos taurus
3.2.1.21 7,8-dideoxy-3-hydroxy-8-octylamino-5-octylimino-6-oxa-3-epi-australine
-
 Prunus dulcis
3.2.1.21 7,8-dideoxy-8-dodecylamino-3-hydroxy-5-octylimino-6-oxa-3-epi-australine
-
 Bos taurus
3.2.1.21 7,8-dideoxy-8-dodecylamino-3-hydroxy-5-octylimino-6-oxa-3-epi-australine
-
 Prunus dulcis
3.2.1.21 8-butylamino-7,8-dideoxy-3-hydroxy-5-octylimino-6-oxa-3-epi-australine
-
 Bos taurus
3.2.1.21 8-butylamino-7,8-dideoxy-3-hydroxy-5-octylimino-6-oxa-3-epi-australine
-
 Prunus dulcis

Organism

EC Number Organism UniProt Comment Textmining
3.2.1.21 Bos taurus
-
-
-
3.2.1.21 Prunus dulcis
-
-
-

Synonyms

EC Number Synonyms Comment Organism
3.2.1.21 beta-Glcase
-
 Bos taurus
3.2.1.21 beta-Glcase
-
 Prunus dulcis

Ki Value [mM]

EC Number Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
3.2.1.21 0.0029
-
 7,8-dideoxy-8-dodecylamino-3-hydroxy-5-octylimino-6-oxa-3-epi-australine pH and temperature not specified in the publication Bos taurus
3.2.1.21 0.0096
-
 7,8-dideoxy-3-hydroxy-8-octylamino-5-octylimino-6-oxa-3-epi-australine pH and temperature not specified in the publication Bos taurus
3.2.1.21 0.012
-
 7,8-dideoxy-3,8-dioctylamino-5-octylimino-6-oxa-3-epi-australine pH and temperature not specified in the publication Bos taurus
3.2.1.21 0.025
-
 7,8-dideoxy-3,8-didodecylamino-5-octylimino-6-oxa-3-epi-australine pH and temperature not specified in the publication Bos taurus
3.2.1.21 0.051
-
 8-butylamino-7,8-dideoxy-3-hydroxy-5-octylimino-6-oxa-3-epi-australine pH and temperature not specified in the publication Bos taurus
3.2.1.21 0.056
-
 7,8-dideoxy-8-dodecylamino-3-hydroxy-5-octylimino-6-oxa-3-epi-australine pH and temperature not specified in the publication Prunus dulcis
3.2.1.21 0.058
-
 3,8-dibutylamino-7,8-dideoxy-5-octylimino-6-oxa-3-epi-australine pH and temperature not specified in the publication Bos taurus
3.2.1.21 0.223
-
 3,8-dibutylamino-7,8-dideoxy-5-octylimino-6-oxa-3-epi-australine pH and temperature not specified in the publication Prunus dulcis
3.2.1.21 0.32
-
 8-butylamino-7,8-dideoxy-3-hydroxy-5-octylimino-6-oxa-3-epi-australine pH and temperature not specified in the publication Prunus dulcis
3.2.1.21 0.367
-
 7,8-dideoxy-3,8-didodecylamino-5-octylimino-6-oxa-3-epi-australine pH and temperature not specified in the publication Prunus dulcis
3.2.1.21 0.441
-
 7,8-dideoxy-3,8-dioctylamino-5-octylimino-6-oxa-3-epi-australine pH and temperature not specified in the publication Prunus dulcis
3.2.1.21 0.484
-
 7,8-dideoxy-3-hydroxy-8-octylamino-5-octylimino-6-oxa-3-epi-australine pH and temperature not specified in the publication Prunus dulcis