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Literature summary extracted from

  • Nachon, F.; Carletti, E.; Ronco, C.; Trovaslet, M.; Nicolet, Y.; Jean, L.; Renard, P.Y.
    Crystal structures of human cholinesterases in complex with huprine W and tacrine: elements of specificity for anti-Alzheimers drugs targeting acetyl- and butyryl-cholinesterase (2013), Biochem. J., 453, 393-399.
    View publication on PubMed

Cloned(Commentary)

EC Number Cloned (Comment) Organism
3.1.1.8 expressed in CHO-K1 cells Homo sapiens

Crystallization (Commentary)

EC Number Crystallization (Comment) Organism
3.1.1.8 in complex with tacrine, hanging drop vapor diffusion method, using 0.1 M MES (pH 6.5) and 2.1 M ammonium sulfate Homo sapiens

Inhibitors

EC Number Inhibitors Comment Organism Structure
3.1.1.8 tacrine
-
Homo sapiens

Organism

EC Number Organism UniProt Comment Textmining
3.1.1.8 Homo sapiens P06276
-
-

Synonyms

EC Number Synonyms Comment Organism
3.1.1.8 BChE
-
Homo sapiens
3.1.1.8 butyrylcholinesterase
-
Homo sapiens