EC Number | Inhibitors | Comment | Organism | Structure |
---|---|---|---|---|
3.4.14.5 | MCB3937 | - |
Homo sapiens | |
3.4.24.11 | MCB3937 | bifunctional inhibitor of NEP and DPP-IV | Homo sapiens | |
3.4.24.11 | MCB4241 | bifunctional inhibitor of NEP and DPP-IV | Homo sapiens | |
3.4.24.11 | thiorphan | - |
Homo sapiens |
EC Number | Organism | UniProt | Comment | Textmining |
---|---|---|---|---|
3.4.14.5 | Homo sapiens | - |
- |
- |
3.4.24.11 | Homo sapiens | P08473 | - |
- |
EC Number | Synonyms | Comment | Organism |
---|---|---|---|
3.4.14.5 | DPP-IV | - |
Homo sapiens |
3.4.24.11 | CALLA | - |
Homo sapiens |
3.4.24.11 | CD10 | - |
Homo sapiens |
3.4.24.11 | enkephalinase | - |
Homo sapiens |
3.4.24.11 | NEP | - |
Homo sapiens |
EC Number | Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|---|
3.4.24.11 | 0.000004 | - |
thiorphan | - |
Homo sapiens |
EC Number | IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|---|
3.4.14.5 | 0.0003 | - |
- |
Homo sapiens | MCB3937 | |
3.4.24.11 | 0.00045 | - |
- |
Homo sapiens | MCB3937 | |
3.4.24.11 | 0.0006 | - |
- |
Homo sapiens | MCB4241 |