EC Number | Inhibitors | Comment | Organism | Structure |
---|---|---|---|---|
1.17.4.4 | warfarin | IC50: 0.00007 mM | Bos taurus | |
1.17.4.4 | warfarin | - |
Canis lupus familiaris | |
1.17.4.4 | warfarin | - |
Equus caballus | |
1.17.4.4 | warfarin | IC50: 0.00018 mM, only one sample measured | Homo sapiens | |
1.17.4.4 | warfarin | IC50: 0.00017 mM | Mus musculus | |
1.17.4.4 | warfarin | - |
Ovis aries | |
1.17.4.4 | warfarin | IC50: 0.00012 mM, only one sample measured | Sus scrofa |
EC Number | KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|---|
1.17.4.4 | 0.00241 | - |
vitamin K1 2,3-epoxide | 37°C | Ovis aries | |
1.17.4.4 | 0.00241 | - |
vitamin K1 2,3-epoxide | 37°C | Equus caballus | |
1.17.4.4 | 0.00309 | - |
vitamin K1 2,3-epoxide | 37°C, only one sample measured | Homo sapiens | |
1.17.4.4 | 0.0032 | - |
vitamin K1 2,3-epoxide | 37°C, only one sample measured | Sus scrofa | |
1.17.4.4 | 0.0036 | - |
vitamin K1 2,3-epoxide | 37°C | Canis lupus familiaris | |
1.17.4.4 | 0.00416 | - |
vitamin K1 2,3-epoxide | 37°C | Mus musculus | |
1.17.4.4 | 0.00425 | - |
vitamin K1 2,3-epoxide | 37°C | Bos taurus | |
1.17.4.4 | 0.00646 | - |
vitamin K1 2,3-epoxide | 37°C | Bos taurus |
EC Number | Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|---|
1.17.4.4 | microsome | - |
Mus musculus | - |
- |
1.17.4.4 | microsome | - |
Homo sapiens | - |
- |
1.17.4.4 | microsome | - |
Sus scrofa | - |
- |
1.17.4.4 | microsome | - |
Bos taurus | - |
- |
1.17.4.4 | microsome | - |
Ovis aries | - |
- |
1.17.4.4 | microsome | - |
Canis lupus familiaris | - |
- |
1.17.4.4 | microsome | - |
Equus caballus | - |
- |
EC Number | Organism | UniProt | Comment | Textmining |
---|---|---|---|---|
1.17.4.4 | Bos taurus | - |
- |
- |
1.17.4.4 | Canis lupus familiaris | - |
- |
- |
1.17.4.4 | Equus caballus | - |
- |
- |
1.17.4.4 | Homo sapiens | - |
- |
- |
1.17.4.4 | Mus musculus | - |
- |
- |
1.17.4.4 | Ovis aries | - |
- |
- |
1.17.4.4 | Sus scrofa | - |
- |
- |
EC Number | Source Tissue | Comment | Organism | Textmining |
---|---|---|---|---|
1.17.4.4 | liver | - |
Mus musculus | - |
1.17.4.4 | liver | - |
Homo sapiens | - |
1.17.4.4 | liver | - |
Sus scrofa | - |
1.17.4.4 | liver | - |
Bos taurus | - |
1.17.4.4 | liver | - |
Ovis aries | - |
1.17.4.4 | liver | - |
Canis lupus familiaris | - |
1.17.4.4 | liver | - |
Equus caballus | - |
EC Number | Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|---|
1.17.4.4 | vitamin K1 2,3-epoxide + dithiothreitol | - |
Mus musculus | vitamin K1 + oxidized dithiothreitol | - |
? | |
1.17.4.4 | vitamin K1 2,3-epoxide + dithiothreitol | - |
Homo sapiens | vitamin K1 + oxidized dithiothreitol | - |
? | |
1.17.4.4 | vitamin K1 2,3-epoxide + dithiothreitol | - |
Sus scrofa | vitamin K1 + oxidized dithiothreitol | - |
? | |
1.17.4.4 | vitamin K1 2,3-epoxide + dithiothreitol | - |
Bos taurus | vitamin K1 + oxidized dithiothreitol | - |
? | |
1.17.4.4 | vitamin K1 2,3-epoxide + dithiothreitol | - |
Ovis aries | vitamin K1 + oxidized dithiothreitol | - |
? | |
1.17.4.4 | vitamin K1 2,3-epoxide + dithiothreitol | - |
Canis lupus familiaris | vitamin K1 + oxidized dithiothreitol | - |
? | |
1.17.4.4 | vitamin K1 2,3-epoxide + dithiothreitol | - |
Equus caballus | vitamin K1 + oxidized dithiothreitol | - |
? |
EC Number | Synonyms | Comment | Organism |
---|---|---|---|
1.17.4.4 | VKOR | - |
Mus musculus |
1.17.4.4 | VKOR | - |
Homo sapiens |
1.17.4.4 | VKOR | - |
Sus scrofa |
1.17.4.4 | VKOR | - |
Bos taurus |
1.17.4.4 | VKOR | - |
Ovis aries |
1.17.4.4 | VKOR | - |
Canis lupus familiaris |
1.17.4.4 | VKOR | - |
Equus caballus |
1.17.4.4 | warfarin-sensitive vitamin K1 2,3-epoxide reductase | - |
Mus musculus |
1.17.4.4 | warfarin-sensitive vitamin K1 2,3-epoxide reductase | - |
Homo sapiens |
1.17.4.4 | warfarin-sensitive vitamin K1 2,3-epoxide reductase | - |
Sus scrofa |
1.17.4.4 | warfarin-sensitive vitamin K1 2,3-epoxide reductase | - |
Bos taurus |
1.17.4.4 | warfarin-sensitive vitamin K1 2,3-epoxide reductase | - |
Ovis aries |
1.17.4.4 | warfarin-sensitive vitamin K1 2,3-epoxide reductase | - |
Canis lupus familiaris |
1.17.4.4 | warfarin-sensitive vitamin K1 2,3-epoxide reductase | - |
Equus caballus |
EC Number | IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|---|
1.17.4.4 | 0.00007 | - |
IC50: 0.00007 mM | Bos taurus | warfarin | |
1.17.4.4 | 0.00012 | - |
IC50: 0.00012 mM, only one sample measured | Sus scrofa | warfarin | |
1.17.4.4 | 0.00017 | - |
IC50: 0.00017 mM | Mus musculus | warfarin | |
1.17.4.4 | 0.00018 | - |
IC50: 0.00018 mM, only one sample measured | Homo sapiens | warfarin |