EC Number | Application | Comment | Organism |
---|---|---|---|
3.4.24.23 | medicine | development of effective inhibitors useful for cancer therapy | Homo sapiens |
EC Number | Cloned (Comment) | Organism |
---|---|---|
3.4.24.23 | recombinant pro-matrilysin | Homo sapiens |
EC Number | Inhibitors | Comment | Organism | Structure |
---|---|---|---|---|
3.4.24.23 | additional information | no inhibition with phosphoramidon | Homo sapiens | |
3.4.24.23 | R-94138 | - |
Homo sapiens | |
3.4.24.23 | thiorphan | - |
Homo sapiens | |
3.4.24.23 | Zincov | - |
Homo sapiens |
EC Number | Organism | UniProt | Comment | Textmining |
---|---|---|---|---|
3.4.24.23 | Homo sapiens | - |
human | - |
EC Number | Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|---|
3.4.24.23 | (7-methoxycoumarin-4-yl)acetyl-L-Pro-L-Leu-Gly-L-Leu-[N3-(2,4-dinitrophenyl)-L-2,3-diamino-propionyl]-L-Ala-L-Arg-NH2 + H2O | MOCAc-PLGL(Dpa)AR, Lot 480429 | Homo sapiens | ? | - |
? |
EC Number | Synonyms | Comment | Organism |
---|---|---|---|
3.4.24.23 | matrilysin | - |
Homo sapiens |
3.4.24.23 | Matrix metalloproteinase 7 | - |
Homo sapiens |
3.4.24.23 | MMP-7 | - |
Homo sapiens |
EC Number | pH Minimum | pH Maximum | Comment | Organism |
---|---|---|---|---|
3.4.24.23 | 4 | 10 | - |
Homo sapiens |
EC Number | Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|---|
3.4.24.23 | 0.0105 | - |
R-94138 | pH 7.5, 25°C | Homo sapiens | |
3.4.24.23 | 0.0112 | - |
thiorphan | pH 7.5, 25°C | Homo sapiens | |
3.4.24.23 | 0.015 | - |
thiorphan | pH 7.5, 37°C | Homo sapiens |