Inhibitors | Comment | Organism | Structure |
---|---|---|---|
bis(maltolato)oxovanadium(IV) | - |
Oryctolagus cuniculus | |
bis(N-hydroxylamidoiminodiacetato)vanadium(IV) | - |
Oryctolagus cuniculus | |
pyridine-2,6-dicarboxylatodioxovanadium | - |
Oryctolagus cuniculus | |
vanadate | - |
Oryctolagus cuniculus |
Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|
sarcoplasmic reticulum | - |
Oryctolagus cuniculus | 16529 | - |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
Ca2+ | dependent on | Oryctolagus cuniculus |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Oryctolagus cuniculus | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
skeletal muscle | - |
Oryctolagus cuniculus | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + H2O + Ca2+/cis | - |
Oryctolagus cuniculus | ADP + phosphate + Ca2+/trans | - |
? |
Synonyms | Comment | Organism |
---|---|---|
sarcoplasmic reticulum calcium ATPase | - |
Oryctolagus cuniculus |
SR Ca2+-ATPase | - |
Oryctolagus cuniculus |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.025 | - |
in 25 mM HEPES (pH 7.0), 100 mM KCl, 5 mM MgCl2, 0.05 mM CaCl2, at 25°C | Oryctolagus cuniculus | pyridine-2,6-dicarboxylatodioxovanadium | |
0.04 | - |
in 25 mM HEPES (pH 7.0), 100 mM KCl, 5 mM MgCl2, 0.05 mM CaCl2, at 25°C | Oryctolagus cuniculus | bis(maltolato)oxovanadium(IV) | |
0.08 | - |
in 25 mM HEPES (pH 7.0), 100 mM KCl, 5 mM MgCl2, 0.05 mM CaCl2, at 25°C | Oryctolagus cuniculus | vanadate | |
0.325 | - |
in 25 mM HEPES (pH 7.0), 100 mM KCl, 5 mM MgCl2, 0.05 mM CaCl2, at 25°C | Oryctolagus cuniculus | bis(N-hydroxylamidoiminodiacetato)vanadium(IV) |