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BRENDA support

Literature summary for 3.4.24.71 extracted from

  • Dibas, A.; Prasanna, G.; Yorio, T.
    Characterization of endothelin-converting enzyme activities in ARPE-19 cells, a human retinal pigmented epithelial cell line (2005), J. Ocul. Pharmacol. Ther., 21, 196-204.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
1,10-phenanthroline 1 mM, inhibition of ECE-1 activity Homo sapiens
additional information acidification to pH 6.4 inhibits plasma membrane ECE activity Homo sapiens
phosphoramidon 0.1 M, 35% inhibition of ECE-1 activity Homo sapiens
thiorphan 1 mM, inhibition of ECE-1 activity Homo sapiens

Localization

Localization Comment Organism GeneOntology No. Textmining
plasma membrane
-
Homo sapiens 5886
-

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
retinal pigment epithelium cell line
-
Homo sapiens
-

Synonyms

Synonyms Comment Organism
ECE-1
-
Homo sapiens
endothelin-converting enzyme-1
-
Homo sapiens