Activating Compound | Comment | Organism | Structure |
---|---|---|---|
DTT | activates enzymatic activity up to 0.1 mM | Homo sapiens |
Cloned (Comment) | Organism |
---|---|
expressed in Escherichia coli as a His-tagged fusion protein | Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
1,10-phenanthroline | total inhibition at 10 mM | Homo sapiens | |
bestatin | significant inhibition | Homo sapiens | |
captopril | - |
Homo sapiens | |
DTT | inhibits enzymatic activity above to 0.1 mM | Homo sapiens | |
EDTA | 90% inhibitiond by EDTA (10 mM) | Homo sapiens | |
JA-2 | - |
Homo sapiens | |
thiorphan | - |
Homo sapiens |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.001 | - |
Abz-GFSPFRQ-EDDnp | pH 7.4, 37°C, 0.1 mM DTT | Homo sapiens |
Localization | Comment | Organism | GeneOntology No. | Textmining |
---|
Molecular Weight [Da] | Molecular Weight Maximum [Da] | Comment | Organism |
---|---|---|---|
78640 | - |
mass spectroscopy | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Purification (Comment) | Organism |
---|---|
affinity chromatography using Ni-Sepharose resin and ion exchange chromatography with a Hi-trap resource Q column | Homo sapiens |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
Abz-GFSPFRQ-EDDnp + H2O | - |
Homo sapiens | Abz-GF + SPFRQ-EDDnp | - |
? | |
Abz-RPPGFSPFRQ-EDDnp + H2O | - |
Homo sapiens | Abz-RPPGF + SPFRQ-EDDnp | - |
? | |
bradykinin + H2O | - |
Homo sapiens | ? | - |
? |
Synonyms | Comment | Organism |
---|---|---|
hMIP | - |
Homo sapiens |
mitochondrial intermediate peptidase | - |
Homo sapiens |
Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|
37 | - |
assay at | Homo sapiens |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
7.4 | - |
assay at | Homo sapiens |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.0015 | - |
thiorphan | pH 7.4, 37°C | Homo sapiens | |
0.007 | - |
JA-2 | pH 7.4, 37°C | Homo sapiens | |
0.057 | - |
captopril | pH 7.4, 37°C | Homo sapiens |
kcat/KM Value [1/mMs-1] | kcat/KM Value Maximum [1/mMs-1] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
40 | - |
Abz-GFSPFRQ-EDDnp | pH 7.4, 37°C, 0.1 mM DTT | Homo sapiens |