Activating Compound | Comment | Organism | Structure |
---|---|---|---|
Trypsin | - |
Mus musculus |
Cloned (Comment) | Organism |
---|---|
expressed in human embryonic kidney 293 cells ATCC 1573 CRL | Mus musculus |
Protein Variants | Comment | Organism |
---|---|---|
F161R | site-directed mutagenesis | Mus musculus |
P228K | site-directed mutagenesis | Mus musculus |
Y199K | site-directed mutagenesis | Mus musculus |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.11 | - |
cholecystokinin 8-sulfate | pH 7.5, 37°C, mutant Y199K | Mus musculus | |
0.23 | - |
cholecystokinin 8-sulfate | pH 7.5, 37°C, mutant F161R | Mus musculus | |
0.29 | - |
cholecystokinin 8-sulfate | pH 7.5, 37°C, mutant P228K | Mus musculus | |
0.44 | - |
gastrin 17 | pH 7.5, 37°C, mutant Y199K | Mus musculus | |
0.49 | - |
cholecystokinin 8-sulfate | pH 7.5, 37°C | Mus musculus |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
Zn2+ | zinc-metalloendopeptidase | Mus musculus |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Mus musculus | - |
mouse | - |
Purification (Comment) | Organism |
---|---|
- |
Mus musculus |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
azocasein + H2O | - |
Mus musculus | ? | - |
? | |
cholecystokinin 8-sulfate + H2O | - |
Mus musculus | ? | - |
? | |
gastrin 17 + H2O | mutant Y199K | Mus musculus | ? | - |
? | |
additional information | orcokinin and gastrin 17 are no substrates | Mus musculus | ? | - |
? |
Synonyms | Comment | Organism |
---|---|---|
meprin metalloproteinase | - |
Mus musculus |
mouse meprin alpha | - |
Mus musculus |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
3.8 | - |
cholecystokinin 8-sulfate | pH 7.5, 37°C, mutant P228K | Mus musculus | |
8.6 | - |
cholecystokinin 8-sulfate | pH 7.5, 37°C | Mus musculus | |
10.8 | - |
gastrin 17 | pH 7.5, 37°C, mutant Y199K | Mus musculus | |
13.4 | - |
cholecystokinin 8-sulfate | pH 7.5, 37°C, mutant F161R | Mus musculus | |
14.2 | - |
cholecystokinin 8-sulfate | pH 7.5, 37°C, mutant Y199K | Mus musculus |