Literature summary for 3.4.21.B10 extracted from

Santos, J.A.; Kondo, M.Y.; Freitas, R.F.; dos Santos, M.H.; Ramalho, T.C.; Assis, D.M.; Juliano, L.; Juliano, M.A.; Puzer, L.
The natural flavone fukugetin as a mixed-type inhibitor for human tissue kallikreins (2016), Bioorg. Med. Chem. Lett., 26, 1485-1489 .

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Inhibitors

Inhibitors	Comment	Organism	Structure
fukugetin	mixed-type inhibitor	Homo sapiens

Organism

Organism	UniProt	Comment	Textmining
Homo sapiens	-	-	-

Substrates and Products (Substrate)

Substrates	Comment Substrates	Organism	Products	Comment (Products)	Rev.	Reac.
Abz-KLRSSQ-EDDnp + H2O	-	Homo sapiens	?	-	?

Synonyms

Synonyms	Comment	Organism
KLK6	isoform	Homo sapiens

IC50 Value

IC50 Value	IC50 Value Maximum	Comment	Organism	Inhibitor	Structure
0.0135	-	at pH 7.5 and 37°C	Homo sapiens	fukugetin

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Release 2023.1 (January 2023)